SCHEMBL8890529

SCHEMBL8890529

CC(C)(C)OC(=O)N1CCC(CCNS(=O)(=O)c2cccc3ccccc23)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 11/20 0.53
KDM4E B2RXH2 1/20 0.50
PKM P14618 1/20 0.50
HTR6 P50406 1/20 0.50
STS P08842 2/20 0.48
CCR8 P51685 1/20 0.48
BRD4 O60885 1/20 0.47
GPR119 Q8TDV5 1/20 0.47
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
HDAC9 Q9UKV0 1/20 0.47
HDAC5 Q9UQL6 1/20 0.47
NPY5R Q15761 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8899787 0.91 TGFBR1 (0.64) TGFBR1KDM4EPKMNPY5R
SCHEMBL8899558 0.84 ACKR3 (0.53) HTR6NPY5R
SCHEMBL6347374 0.82 SLC6A9 (0.51) NPY5R
SCHEMBL16112711 0.78 KDM4E (0.58) TGFBR1KDM4EPKMSTSGPR119
SCHEMBL8901280 0.78 TGFBR1 (0.64) TGFBR1KDM4EPKMSTS
SCHEMBL27900155 0.77 SCN1A (0.49) KDM4ENPY5R
SCHEMBL4266289 0.77 CNR1 (0.59) KDM4EHDAC3HDAC4HDAC1HDAC7
SCHEMBL13932868 0.76 HTR2A (0.52) STSGPR119
SCHEMBL2459419 0.75 KDM4E (0.52) TGFBR1KDM4EPKMHTR6GPR119
SCHEMBL14834135 0.75 MGLL (0.64) TGFBR1NPY5R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997020820-A1 HETEROARYL COMPOUNDS NOVARTIS AG (CH) 1997-06-12 WO disclosed