SCHEMBL8899879

SCHEMBL8899879

O=C1C2=C(C(=O)c3ccccc31)C(O)OC(C(=O)C1CC3C(=O)c4ccccc4C(=O)C3=C(O)O1)C2

nearest known ligand 0.33

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AKT1 P31749 5/20 0.33
DNMT3B Q9UBC3 1/20 0.30
HSP90AA1 P07900 1/20 0.30
PAX8 Q06710 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8899885 0.84 AKT1 (0.40) AKT1DNMT3BHSP90AA1PAX8
SCHEMBL8531494 0.68 DNMT3B (0.53) AKT1DNMT3BHSP90AA1PAX8
SCHEMBL8531103 0.66 DNMT3B (0.48) AKT1DNMT3BHSP90AA1PAX8
SCHEMBL8900149 0.63 AKT1 (0.34) AKT1
SCHEMBL8587198 0.62 TCF4 (0.39) AKT1DNMT3BHSP90AA1PAX8
SCHEMBL8900155 0.61 AKT1 (0.47) AKT1
SCHEMBL9755762 0.60 HTT (0.34)
SCHEMBL8900228 0.60 TCF4 (0.39) AKT1DNMT3BHSP90AA1PAX8
SCHEMBL8899620 0.58 AKT1 (0.50) AKT1DNMT3BHSP90AA1PAX8
SCHEMBL8907639 0.57 CTH (0.38) AKT1DNMT3BHSP90AA1PAX8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5606037-A Processes antineoplastic heteronaphthoquinones BIOCHEM PHARMA INC. (CA) 1997-02-25 US claimed
EP-0659190-A1 ANTINEOPLASTIC HETERONAPHTHOQUINONES BIOCHEM PHARMA INC (CA) 1995-06-28 EP claimed
WO-1994011382-A1 ANTINEOPLASTIC HETERONAPHTHOQUINONES BIOCHEM PHARMA INC. (CA) 1994-05-26 WO claimed
US-5606037-A Processes antineoplastic heteronaphthoquinones BIOCHEM PHARMA INC. (CA) 1997-02-25 US disclosed
EP-0659190-A1 ANTINEOPLASTIC HETERONAPHTHOQUINONES BIOCHEM PHARMA INC (CA) 1995-06-28 EP disclosed
WO-1994011382-A1 ANTINEOPLASTIC HETERONAPHTHOQUINONES BIOCHEM PHARMA INC. (CA) 1994-05-26 WO disclosed