SCHEMBL8901086

SCHEMBL8901086

COc1cc(NC(=O)c2ccccc2Cl)ccc1C(=O)N1c2ccc(Cl)cc2C(N2CCN(CCO)CC2)CCC1C=C=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 3/20 0.40
CHRM5 P08912 2/20 0.40
CHRM3 P20309 2/20 0.40
HSD17B10 Q99714 1/20 0.40
AVPR2 P30518 7/20 0.39
GRM4 Q14833 4/20 0.38
ALDH1A1 P00352 2/20 0.38
KMT2A Q03164 2/20 0.38
KDM4E B2RXH2 1/20 0.38
AVPR1A P37288 2/20 0.37
ABCB11 O95342 1/20 0.37
ADRB2 P07550 1/20 0.37
HTR1A P08908 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
TBXA2R P21731 1/20 0.37
HTR2C P28335 1/20 0.37
HRH1 P35367 1/20 0.37
OPRM1 P35372 1/20 0.37
GLP1R P43220 1/20 0.37
TMEM97 Q5BJF2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8900831 0.91 CHRM1 (0.42) CHRM1CHRM5CHRM3HSD17B10AVPR2
SCHEMBL4743947 0.84 GRM4 (0.39) CHRM1CHRM5CHRM3HSD17B10AVPR2
SCHEMBL8634459 0.83 CHRM5 (0.40) CHRM1CHRM5CHRM3HSD17B10AVPR2
SCHEMBL4684270 0.81 AVPR2 (0.41) CHRM1CHRM5CHRM3AVPR2GRM4
SCHEMBL4684920 0.75 AVPR2 (0.48) CHRM1CHRM5CHRM3AVPR2GRM4
SCHEMBL4684917 0.75 AVPR2 (0.49) CHRM1CHRM5CHRM3AVPR2GRM4
SCHEMBL8635111 0.74 CHRM5 (0.41) CHRM1CHRM5CHRM3HSD17B10AVPR2
SCHEMBL7334875 0.73 GRM4 (0.45) CHRM1HSD17B10AVPR2GRM4ALDH1A1
SCHEMBL4682920 0.73 HSD17B10 (0.43) CHRM1CHRM5CHRM3HSD17B10AVPR2
SCHEMBL8630909 0.72 HSD17B10 (0.37) CHRM1CHRM5CHRM3HSD17B10AVPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5622947-A VASODILATORS, HYPOTENSIVE AGENTS, DIURETICS, PLATELET AGGLUTINATION INHIBITORS; ALSO USED TO PREVENT PREMATURE BIRTH, TREAT DYSMENORRHEA OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1997-04-22 US disclosed