SCHEMBL8901284

SCHEMBL8901284

COC(=O)C(O)c1ccc(NCCN(CC(O[Si](C)(C)C(C)(C)C)c2cccc(Cl)c2)C(=O)OC(C)(C)C)cc1

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 8/20 0.33
ADRB1 P08588 7/20 0.33
ADRB2 P07550 6/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
BACE1 P56817 3/20 0.32
AOC3 Q16853 1/20 0.32
LDHA P00338 1/20 0.30
LDHB P07195 1/20 0.30
S1PR3 Q99500 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7714567 0.83 ADRB2 (0.31) ADRB3ADRB1ADRB2
SCHEMBL8100555 0.83 ADRB2 (0.31) ADRB3ADRB1ADRB2
SCHEMBL6432465 0.82 ADRB3 (0.52) ADRB3ADRB1ADRB2
SCHEMBL6432460 0.82 ADRB3 (0.52) ADRB3ADRB1ADRB2
SCHEMBL7714681 0.82 NR1H2 (0.34) ADRB3ADRB1ADRB2
SCHEMBL7714678 0.82 NR1H2 (0.34) ADRB3ADRB1ADRB2
SCHEMBL7716904 0.82 AOC3 (0.36) ADRB3ADRB1ADRB2MEN1KMT2A
SCHEMBL6436830 0.81 ADRB1 (0.42) ADRB3ADRB1ADRB2BACE1
SCHEMBL6436884 0.80 MCHR1 (0.40) ADRB3ADRB1ADRB2
SCHEMBL6436877 0.80 MCHR1 (0.40) ADRB3ADRB1ADRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1997021666-A1 ARYLETHANOLAMINE DERIVATIVES AND THEIR USE AS AGONISTS OF ATYPICAL BETA-ADRENOCEPTORS GLAXO GROUP LIMITED (GB) 1997-06-19 WO disclosed