SCHEMBL8901705

SCHEMBL8901705

O=C1CC[C@@H]([N+](=O)[O-])[C@H](c2ccccc2C(F)(F)F)N1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.67
GAA P10253 1/20 0.67
ATM Q13315 1/20 0.60
ALDH1A1 P00352 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
KMT2A Q03164 5/20 0.51
MEN1 O00255 4/20 0.51
TDP1 Q9NUW8 2/20 0.51
POLB P06746 2/20 0.51
HTR2C P28335 2/20 0.43
DDB1 Q16531 1/20 0.39
CRBN Q96SW2 1/20 0.39
HPN P05981 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
ADORA3 P0DMS8 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4919831 0.81 ATM (0.69) RAB9AGAAATMALDH1A1SMN1; SMN2
SCHEMBL4919848 0.81 ATM (0.69) RAB9AGAAATMALDH1A1SMN1; SMN2
SCHEMBL4919841 0.81 ATM (0.69) RAB9AGAAATMALDH1A1SMN1; SMN2
SCHEMBL5748309 0.80 RAB9A (0.71) RAB9AGAAATMALDH1A1SMN1; SMN2
SCHEMBL9024919 0.80 GAA (1.00) RAB9AGAAATMALDH1A1SMN1; SMN2
SCHEMBL5748304 0.80 RAB9A (0.71) RAB9AGAAATMALDH1A1SMN1; SMN2
SCHEMBL5748307 0.80 RAB9A (0.71) RAB9AGAAATMALDH1A1SMN1; SMN2
SCHEMBL6098746 0.76 SMN1; SMN2 (0.74) RAB9AGAAATMALDH1A1SMN1; SMN2
SCHEMBL7898746 0.76 SMN1; SMN2 (0.74) RAB9AGAAATMALDH1A1SMN1; SMN2
SCHEMBL7898749 0.76 SMN1; SMN2 (0.74) RAB9AGAAATMALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5703240-A ANALGESICS; ANTIINFLAMMATORY AGENTS; NERVOUS SYSTEM DISORDERS; PSYCHOLOGICAL DISORDERS; GASTROINTESTINAL DISORDERS GLAXO GROUP LIMITED (GB) 1997-12-30 US disclosed
EP-0720609-A1 3-(5-TETRAZOLYL-BENZYL)AMINO-PIPERIDINE DERIVATIVES AND ANTAGONISTS OF TACHYKININS GLAXO GROUP LIMITED (GB) 1996-07-10 EP disclosed
WO-1995008549-A1 3-(5-TETRAZOLYL-BENZYL)AMINO-PIPERIDINE DERIVATIVES AND ANTAGONISTS OF TACHYKININS GLAXO GROUP LIMITED (GB) 1995-03-30 WO disclosed