SCHEMBL8903379

SCHEMBL8903379

CC(C)(C)c1cc(-c2nc(OCc3ccc(C(=O)O)cc3)c3[nH]cnc3n2)cc(C(C)(C)C)c1O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 7/20 0.43
RXRA P19793 3/20 0.43
RXRB P28702 3/20 0.43
RXRG P48443 2/20 0.43
MGMT P16455 5/20 0.43
CDK1 P06493 2/20 0.43
CCNB1 P14635 2/20 0.43
CCNA2 P20248 2/20 0.43
CDK2 P24941 2/20 0.43
CCNA1 P78396 2/20 0.43
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
TSHR P16473 1/20 0.43
NFKB1 P19838 1/20 0.43
CYP2C19 P33261 1/20 0.43
BLM P54132 1/20 0.43
PMP22 Q01453 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8903375 0.85 RXRA (0.43) RXRARXRBRXRGNR4A2GAA
SCHEMBL8903387 0.81 CDK1 (0.39) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL8902502 0.80 CDK1 (0.55) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL8901822 0.79 PTGS2 (0.46)
SCHEMBL8903318 0.79 CDK1 (0.53) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL8901655 0.77 CDK1 (0.55) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL8902911 0.77 CDK1 (0.55) PIN1MGMTCDK1CCNB1CCNA2
SCHEMBL8902849 0.76 CA1 (0.43)
SCHEMBL8903481 0.73 DAPK1 (0.45) RXRARXRBRXRGGAAMAPT
SCHEMBL9854008 0.73 RXRA (0.63) RXRARXRBRXRGTSHRNR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5602140-A CAUSED BY LEUKOCYTES JAPAN ENERGY CORPORATION (JP) 1997-02-11 US disclosed
EP-0675124-A2 Purine derivatives and suppressants for inflammatory diseases JAPAN ENERGY CORPORATION (JP) 1995-10-04 EP disclosed