SCHEMBL8903167

SCHEMBL8903167

CC1(C)CCN(C(=O)CI)CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.37
ALDH1A1 P00352 5/20 0.33
EPHX2 P34913 1/20 0.33
L3MBTL1 Q9Y468 2/20 0.32
ATM Q13315 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
USP2 O75604 1/20 0.32
LMNA P02545 1/20 0.32
CYP3A4 P08684 1/20 0.32
HPGD P15428 1/20 0.32
KMT2A Q03164 1/20 0.32
HSD17B10 Q99714 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
SPR P35270 1/20 0.32
NPC1 O15118 1/20 0.31
CYP1A2 P05177 1/20 0.31
JAK2 O60674 1/20 0.31
JAK1 P23458 1/20 0.31
JAK3 P52333 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13360768 0.80 ALDH1A1 (0.52) NAMPTALDH1A1EPHX2L3MBTL1MEN1
SCHEMBL14417828 0.80 NAMPT (0.42) NAMPTALDH1A1EPHX2L3MBTL1ATM
SCHEMBL13438125 0.78 CPN1 (0.39) NAMPTALDH1A1EPHX2ATMKDM4E
SCHEMBL14417834 0.78 NAMPT (0.37) NAMPTALDH1A1EPHX2L3MBTL1ATM
SCHEMBL13194913 0.78 ALDH1A1 (0.41) NAMPTALDH1A1EPHX2L3MBTL1ATM
SCHEMBL4438715 0.78 ALDH1A1 (0.53) NAMPTALDH1A1LMNASPR
SCHEMBL9275712 0.78 ALDH1A1 (0.48) ALDH1A1L3MBTL1ATMKDM4EMEN1
SCHEMBL8903212 0.78 ALDH1A1 (0.40) ALDH1A1L3MBTL1ATMKDM4EMEN1
SCHEMBL13194846 0.78 OPRM1 (0.35) NAMPTALDH1A1OPRM1
SCHEMBL8904836 0.77 ALDH1A1 (0.41) ALDH1A1ATMUSP2CYP3A4HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5618808-A Benzothiazepine and benzoxazepine derivatives as cholecystokinin receptor antagonists PFIZER, INC. (US) 1997-04-08 US disclosed
EP-0648213-A1 BENZOTHIAZEPINE AND BENZOXAZEPINE DERIVATIVES AS CHOLECYSTOKININ RECEPTOR ANTAGONISTS PFIZER INC. (US) 1995-04-19 EP disclosed
WO-1994001421-A1 BENZOTHIAZEPINE AND BENZOXAZEPINE DERIVATIVES AS CHOLECYSTOKININ RECEPTOR ANTAGONISTS PFIZER INC. (US) 1994-01-20 WO disclosed