SCHEMBL8903418

SCHEMBL8903418

Cc1oc(C(=O)NC2CCC(OCC(=O)OC(C)(C)C)CC2)c2ccc(C#N)cc12

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.38
CETP P11597 8/20 0.38
ABCB1 P08183 1/20 0.36
IRAK4 Q9NWZ3 1/20 0.35
EGLN1 Q9GZT9 2/20 0.34
KDM1A O60341 2/20 0.34
PDE4B Q07343 2/20 0.33
PDE4A P27815 1/20 0.33
PDE4C Q08493 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KCNH2 Q12809 1/20 0.33
MCHR1 Q99705 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8904770 0.90 CETP (0.37) DRD2CETPABCB1IRAK4EGLN1
SCHEMBL8905478 0.87 NPC1 (0.46) CETPNPC1RAB9AMCHR1
SCHEMBL8716441 0.87 NPC1 (0.46) CETPNPC1RAB9AMCHR1
SCHEMBL8904014 0.85 DRD2 (0.39) DRD2CETPABCB1IRAK4PDE4B
SCHEMBL8904764 0.84 CETP (0.40) DRD2CETPABCB1IRAK4NPC1
SCHEMBL8713211 0.84 CETP (0.40) DRD2CETPABCB1IRAK4NPC1
SCHEMBL8906283 0.83 ITGB3 (0.40)
SCHEMBL8715642 0.80 CETP (0.43) DRD2CETPABCB1NPC1RAB9A
SCHEMBL8904008 0.80 CETP (0.43) DRD2CETPABCB1NPC1RAB9A
SCHEMBL8713035 0.77 DRD2 (0.49) DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5635527-A ANTAGONIST OF PLATELET MEMBRANE GLYCOPROTEIN; TREATMENT OF THROMBOTIC DISEASES THE GREEN CROSS CORPORATION (JP) 1997-06-03 US disclosed
EP-0712844-A1 NOVEL FUSED-RING CARBOXYLIC ACID COMPOUND OR SALT THEREOF, AND MEDICINAL USE THEREOF THE GREEN CROSS CORPORATION (JP) 1996-05-22 EP disclosed