SCHEMBL8904346

SCHEMBL8904346

CC1CC(=O)c2cccc(C(N)=S)c21

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.36
ACHE P22303 3/20 0.35
KEAP1 Q14145 1/20 0.32
NFE2L2 Q16236 1/20 0.32
STAT3 P40763 1/20 0.31
S100A4 P26447 1/20 0.31
NOTUM Q6P988 2/20 0.30
CSNK2A2 P19784 1/20 0.30
CSNK2A1 P68400 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8903529 0.83 PARP1 (0.35) PARP1ACHEKEAP1NFE2L2STAT3
SCHEMBL8903467 0.75 ACHE (0.57) PARP1ACHEKEAP1NFE2L2STAT3
SCHEMBL2480306 0.73 ACHE (0.41) ACHESTAT3S100A4CSNK2A2CSNK2A1
SCHEMBL8734160 0.69 ACHE (0.38) ACHESTAT3S100A4CSNK2A2CSNK2A1
SCHEMBL6812230 0.68 PARP1 (0.40) PARP1KEAP1NFE2L2
SCHEMBL8903475 0.68 ACHE (0.40) ACHES100A4
SCHEMBL6808475 0.66 BRD4 (0.45) PARP1KEAP1NFE2L2
SCHEMBL181579 0.63 ACHE (0.48) ACHES100A4NOTUMCSNK2A2CSNK2A1
SCHEMBL9367273 0.63 ACHE (0.48) ACHES100A4NOTUMCSNK2A2CSNK2A1
SCHEMBL9372008 0.63 ACHE (0.48) ACHES100A4NOTUMCSNK2A2CSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5639911-A Hydrazones CIBA-GEIGY CORPORATION (US) 1997-06-17 US disclosed
US-5461076-A Inhibitors of S-adenosylmethionine decarboxylase; antitumor agents NOVARTIS CORPORATION 1995-10-24 US disclosed
EP-0456133-B1 Hydrazones CIBA GEIGY AG (CH) 1995-03-15 EP disclosed
US-5395855-A Antitumor agents CIBA-GEIGY CORPORATION (US) 1995-03-07 US disclosed
EP-0538193-A2 Condensed cycloaliphatir-amidino-hydrazon salts as S-adenosylmethionin decarboxylase inhibitors CIBA-GEIGY AG (CH) 1993-04-21 EP disclosed
EP-0456133-A1 Hydrazones CIBA-GEIGY AG (CH) 1991-11-13 EP disclosed