SCHEMBL8905641

SCHEMBL8905641

CCCOc1ccc(C(=O)c2ccc(Cc3ccc(=O)[nH]n3)n2C)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.40
CYP19A1 P11511 2/20 0.39
ALOX15 P16050 2/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
ALDH1A1 P00352 4/20 0.37
MAPT P10636 4/20 0.37
LMNA P02545 3/20 0.37
HTT P42858 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CXCL8 P10145 1/20 0.37
AKR1B1 P15121 1/20 0.37
PTGS1 P23219 1/20 0.37
PTGS2 P35354 1/20 0.37
GLO1 Q04760 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
KDM4E B2RXH2 2/20 0.37
HPGD P15428 2/20 0.37
KMT2A Q03164 1/20 0.37
POLB P06746 1/20 0.36
THRB P10828 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8904746 0.92 NPSR1 (0.41) PLK1ALOX15L3MBTL1ALDH1A1MAPT
SCHEMBL8905554 0.87 LMNA (0.45) ALOX15L3MBTL1ALDH1A1MAPTLMNA
SCHEMBL8905744 0.84 CXCL8 (0.38) ALOX15ALDH1A1MAPTLMNAHTT
SCHEMBL8904821 0.84 CXCL8 (0.41) PLK1ALOX15ALDH1A1MAPTLMNA
SCHEMBL8905800 0.84 AKR1B1 (0.54) L3MBTL1ALDH1A1MAPTLMNASMN1; SMN2
SCHEMBL8904190 0.83 AKR1B1 (0.41) ALDH1A1MAPTLMNASMN1; SMN2CXCL8
SCHEMBL8905896 0.83 PTGS2 (0.41) ALDH1A1LMNAHTTSMN1; SMN2CXCL8
SCHEMBL8905930 0.83 AKR1B1 (0.41) LMNASMN1; SMN2CXCL8AKR1B1PTGS1
SCHEMBL8904844 0.82 AKR1B1 (0.43) ALDH1A1MAPTLMNASMN1; SMN2CXCL8
SCHEMBL8904295 0.82 CXCL8 (0.39) CXCL8AKR1B1PTGS1PTGS2GLO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5622948-A ANALGESICS SYNTEX (U.S.A.) INC. (US) 1997-04-22 US disclosed
EP-0714895-A1 Pyrrole derivatives F. Hoffmann-La Roche AG (CH) 1996-06-05 EP disclosed