SCHEMBL8906963

SCHEMBL8906963

Cn1c(C(F)(F)F)c(-c2cc(F)c(C#N)cc2F)c(=O)[nH]c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
TRPV4 Q9HBA0 1/20 0.35
GAA P10253 3/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
BCAT2 O15382 6/20 0.33
BCAT1 P54687 6/20 0.33
DRD2 P14416 1/20 0.32
DRD3 P35462 1/20 0.32
PGR P06401 2/20 0.32
KDM4E B2RXH2 2/20 0.32
ALDH1A1 P00352 2/20 0.32
GLA P06280 2/20 0.32
HPGD P15428 2/20 0.32
AR P10275 2/20 0.32
TP53 P04637 1/20 0.32
PDE4A P27815 1/20 0.32
PDE4B Q07343 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6984955 0.91 BCAT2 (0.36) L3MBTL1MEN1KMT2AGAASMN1; SMN2
SCHEMBL7010249 0.90 KMT2A (0.36) L3MBTL1MEN1KMT2AGAASMN1; SMN2
SCHEMBL8381949 0.90 L3MBTL1 (0.34) L3MBTL1MEN1KMT2AGAASMN1; SMN2
SCHEMBL8594988 0.90 L3MBTL1 (0.34) L3MBTL1MEN1KMT2AGAASMN1; SMN2
SCHEMBL9023675 0.88 TRPV4 (0.33) TRPV4GAABCAT2BCAT1PGR
SCHEMBL7499497 0.88 L3MBTL1 (0.33) L3MBTL1MEN1KMT2AGAASMN1; SMN2
SCHEMBL7030310 0.88 L3MBTL1 (0.40) L3MBTL1GAABCAT2BCAT1PGR
SCHEMBL8541763 0.88 GAA (0.34) L3MBTL1MEN1KMT2AGAASMN1; SMN2
SCHEMBL7026368 0.87 RET (0.37) L3MBTL1KMT2ASMN1; SMN2TDP1BCAT2
SCHEMBL6987528 0.87 SMN1; SMN2 (0.32) L3MBTL1MEN1KMT2AGAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0759908-A1 SUBSTITUTED DIAZACYCLOHEXANDI(THI)ONES BAYER AG (DE) 1997-03-05 EP disclosed
WO-1995031440-A1 SUBSTITUTED DIAZACYCLOHEXANDI(THI)ONES BAYER AKTIENGESELLSCHAFT (DE) 1995-11-23 WO disclosed