SCHEMBL8907232

SCHEMBL8907232

CCCc1nc2ccc(NCS(=O)(=O)c3ccccc3)cc2n1-c1ccc(-c2ccccc2)c(-c2nnn[nH]2)c1C

nearest known ligand 0.32

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.31
CYP2C9 P11712 2/20 0.31
CYP1A2 P05177 2/20 0.31
CYP2C19 P33261 1/20 0.31
RORC P51449 1/20 0.30
CYP2D6 P10635 1/20 0.30
ALDH1A1 P00352 1/20 0.30
THRB P10828 1/20 0.30
HPGD P15428 1/20 0.30
PDE10A Q9Y233 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8906329 0.95 CYP1A2 (0.33) CYP3A4CYP2C9CYP1A2CYP2C19
SCHEMBL8905588 0.82 PPARG (0.35) RORCALDH1A1THRBHPGD
SCHEMBL8905804 0.80 KDM4E (0.40) CYP3A4CYP2C9ALDH1A1HPGD
SCHEMBL8905647 0.78 CYP1A2 (0.33) CYP1A2HPGDPDE10A
SCHEMBL8905446 0.78 AGTR1 (0.38)
SCHEMBL8789960 0.78 PPARG (0.47)
SCHEMBL8907533 0.77 CYP3A4 (0.34) CYP3A4CYP2C9CYP1A2CYP2C19PDE10A
SCHEMBL8906651 0.77 GPR119 (0.38)
SCHEMBL8905214 0.77 PPARG (0.37) CYP3A4CYP2C9ALDH1A1
SCHEMBL8906188 0.76 PDE4A (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5684029-A HYPOTENSIVE AGENTS KARL THOMAE GMBH (DE) 1997-11-04 US disclosed