SCHEMBL8907794

SCHEMBL8907794

CCCc1c(C=O)ccc(C(C)(C)C)c1O[SiH](C)C

nearest known ligand 0.31

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CYSLTR2 Q9NS75 1/20 0.31
CYSLTR1 Q9Y271 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1620797 0.83 ALDH1A1 (0.34)
SCHEMBL5383978 0.78 CA1 (0.39)
SCHEMBL1620557 0.78 CA1 (0.39)
SCHEMBL1010833 0.74 CA2 (0.41)
SCHEMBL7342226 0.74 PPARG (0.31)
SCHEMBL28654089 0.72 ALOX12 (0.37)
SCHEMBL8405501 0.70
SCHEMBL8700619 0.70 CA2 (0.33)
SCHEMBL4580139 0.68
SCHEMBL8126043 0.68 CA1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686478-A Endothelin antagonists MERCK & CO. INC. (US) 1997-11-11 US disclosed
EP-0710235-A4 1996-06-12 EP disclosed
EP-0710235-A1 ENDOTHELIN ANTAGONISTS MERCK & CO. INC. (US) 1996-05-08 EP disclosed
WO-1995003295-A1 ENDOTHELIN ANTAGONISTS MERCK & CO., INC. (US) 1995-02-02 WO disclosed