SCHEMBL8908156

SCHEMBL8908156

COc1cc(-c2c(C(F)(F)F)n(C)c(=O)[nH]c2=O)c(Cl)cc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 2/20 0.43
BCAT1 P54687 2/20 0.43
ALDH1A1 P00352 3/20 0.37
KDM4E B2RXH2 2/20 0.37
HPGD P15428 2/20 0.37
THRB P10828 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
CYP2C9 P11712 1/20 0.33
SUV39H2 Q9H5I1 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
HSP90AA1 P07900 4/20 0.33
HSP90AB1 P08238 3/20 0.33
MAPT P10636 2/20 0.33
NPSR1 Q6W5P4 2/20 0.33
PKM P14618 1/20 0.33
MAPK1 P28482 1/20 0.33
RAB9A P51151 1/20 0.33
CCR6 P51684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8418727 0.80 SMN1; SMN2 (0.39) BCAT2BCAT1ALDH1A1KDM4EHPGD
SCHEMBL7030310 0.76 L3MBTL1 (0.40) BCAT2BCAT1ALDH1A1KDM4EGLA
SCHEMBL8687627 0.74 DRD1 (0.31) DRD1
SCHEMBL30940103 0.74 KMO (0.32) DRD1
SCHEMBL9312250 0.73 KMO (0.32)
SCHEMBL7488864 0.73 SMN1; SMN2 (0.36) BCAT2BCAT1ALDH1A1KDM4EHPGD
SCHEMBL6219513 0.71 GRIK1 (0.33) ALDH1A1KMT2A
SCHEMBL8784413 0.71 BRD4 (0.32) DRD1
SCHEMBL6217982 0.71 LMNA (0.31) KMT2A
SCHEMBL2590560 0.70 BCAT2 (0.34) BCAT2BCAT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0759908-A1 SUBSTITUTED DIAZACYCLOHEXANDI(THI)ONES BAYER AG (DE) 1997-03-05 EP disclosed
WO-1995031440-A1 SUBSTITUTED DIAZACYCLOHEXANDI(THI)ONES BAYER AKTIENGESELLSCHAFT (DE) 1995-11-23 WO disclosed