SCHEMBL8908784

SCHEMBL8908784

COC(=O)C(C)N(C(=O)OC(C)(C)C)C1CCC(=O)CC1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.38
TSHR P16473 1/20 0.35
CA12 O43570 1/20 0.34
CA14 Q9ULX7 1/20 0.34
MT-CO2 P00403 1/20 0.33
NFKB1 P19838 2/20 0.32
NFKB2 Q00653 2/20 0.32
RELA Q04206 2/20 0.32
DDB1 Q16531 1/20 0.30
CRBN Q96SW2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8908787 1.00 THRB (0.38) THRBTSHRCA12CA14MT-CO2
SCHEMBL6139102 0.89 CA14 (0.39) THRBTSHRCA12CA14NFKB1
SCHEMBL9800648 0.87 MT-CO2 (0.32) MT-CO2NFKB1NFKB2RELADDB1
SCHEMBL9800650 0.87 MT-CO2 (0.32) MT-CO2NFKB1NFKB2RELADDB1
SCHEMBL6294190 0.85 TSHR (0.47) THRBTSHRCA12CA14
SCHEMBL7272503 0.85 TSHR (0.47) THRBTSHRCA12CA14
SCHEMBL8910731 0.83 CA12 (0.38) TSHRCA12CA14
SCHEMBL8909370 0.81 CA12 (0.34) TSHRCA12CA14
SCHEMBL8909366 0.81 CA12 (0.34) TSHRCA12CA14
SCHEMBL24969074 0.75 NFKB1 (0.41) MT-CO2NFKB1NFKB2RELADDB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5688946-A DIPEPTIDES FOR HYPOTENSIVE AGENTS AND CARDIOVASCULAR DISORDERS HOFFMANN LA ROCHE INC. (US) 1997-11-18 US disclosed