SCHEMBL8908923

SCHEMBL8908923

O=C(Cc1ccccc1)OC1CCNCC1

nearest known ligand 0.54

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 5/20 0.53
HRH1 P35367 5/20 0.51
CHRM3 P20309 1/20 0.48
ALDH1A1 P00352 1/20 0.46
MAPK1 P28482 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
GBA1 P04062 1/20 0.46
PAM P19021 1/20 0.45
STS P08842 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6761969 0.85 CYP19A1 (0.66) CYP19A1ALDH1A1MAPK1L3MBTL1PAM
SCHEMBL5049441 0.85 CYP19A1 (0.71) CYP19A1ALDH1A1MAPK1L3MBTL1PAM
SCHEMBL5048395 0.84 CYP19A1 (0.75) CYP19A1
SCHEMBL27820726 0.83 CYP19A1 (0.71) CYP19A1ALDH1A1MAPK1L3MBTL1PAM
SCHEMBL1301606 0.83 CYP19A1 (0.71) CYP19A1ALDH1A1MAPK1L3MBTL1PAM
Hydrochloric Acid SCHEMBL4072239 0.83 TDP1 (0.50) HRH1CHRM3GBA1
SCHEMBL27280787 0.82 CYP19A1 (0.54) CYP19A1ALDH1A1MAPK1L3MBTL1PAM
SCHEMBL29099957 0.81 CYP19A1 (0.53) CYP19A1ALDH1A1MAPK1L3MBTL1PAM
SCHEMBL13266074 0.78 ALDH1A1 (0.64) CYP19A1HRH1CHRM3ALDH1A1
SCHEMBL3357147 0.78 MGLL (0.52) CHRM3ALDH1A1MAPK1L3MBTL1GBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101959882-A Imidazole carbonyl compound DAIICHI SANKYO CO LTD 2011-01-26 CN disclosed
CN-101454299-A Ureide derivative and use thereof for medical purposes TORAY INDUSTRIES (JP) 2009-06-10 CN disclosed
CN-1150192-C Piperidines as CCR5 modulators 2004-05-19 CN disclosed
CN-1331691-A Piperidines as CCR5 modulators PFIZER LTD (US) 2002-01-16 CN disclosed
CN-1183770-A Piperazine derivatives, medicaments containing these compounds, their use and processes for their preparation THOMAE GMBH DR K (DE) 1998-06-03 CN disclosed
US-5661148-A ANTIHYPOXIC AGENT FOR RESPIRATORY SYSTEM DISORDER TEIJIN LIMITED (JP) 1997-08-26 US disclosed
EP-0514540-B1 PYRROLO 2,3-d]PYRIMIDINE DERIVATIVE, PROCESS FOR PREPARING THE SAME, AND PHARMACEUTICAL PREPARATION COMPRISING THE DERIVATIVE AS ACTIVE INGREDIENT TEIJIN LTD (JP) 1996-07-17 EP disclosed
EP-0514540-A1 PYRROLO 2,3-d]PYRIMIDINE DERIVATIVE, PROCESS FOR PREPARING THE SAME, AND PHARMACEUTICAL PREPARATION COMPRISING THE DERIVATIVE AS ACTIVE INGREDIENT TEIJIN LIMITED (JP) 1992-11-25 EP disclosed