SCHEMBL8908949

SCHEMBL8908949

NS(=O)(=O)c1cc(-c2ccc(F)c(F)c2)c(-c2ncco2)cc1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 5/20 0.40
FEN1 P39748 5/20 0.40
KIF11 P52732 3/20 0.38
CFTR P13569 1/20 0.38
NR1H2 P55055 2/20 0.37
NR1H3 Q13133 2/20 0.37
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
CA5B Q9Y2D0 1/20 0.36
PTGS2 P35354 5/20 0.35
PTGS1 P23219 4/20 0.35
PDE3B Q13370 1/20 0.35
PDE3A Q14432 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8551071 0.85 NTRK1 (0.41) CFTRNR1H2NR1H3CA12CA1
SCHEMBL8554062 0.70 CA1 (0.44) CA12CA1CA2CA4CA7
SCHEMBL8908994 0.68 MAOB (0.47) CA12CA1CA2CA4CA7
SCHEMBL6026444 0.65 BRD4 (0.43) ALOX5APFEN1CA12CA1CA2
SCHEMBL6728769 0.65 FEN1 (0.46) ALOX5APFEN1CA1CA2PTGS2
SCHEMBL8659162 0.65 KIF11 (0.55) ALOX5APFEN1KIF11PTGS2PTGS1
SCHEMBL8663462 0.65 ALOX5AP (0.46) ALOX5APFEN1KIF11PTGS2PTGS1
SCHEMBL6986037 0.63 EDNRB (0.56) ALOX5APFEN1
SCHEMBL6724115 0.63 KIF11 (0.78) KIF11PTGS2PTGS1
SCHEMBL18230068 0.63 PIK3CD (0.40) ALOX5APFEN1NR1H2NR1H3PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5700816-A ANTIARTHRITIC AGENTS G.D. SEARLE & CO. 1997-12-23 US claimed
US-5700816-A ANTIARTHRITIC AGENTS G.D. SEARLE & CO. 1997-12-23 US disclosed