SCHEMBL8908994

SCHEMBL8908994

Cc1cc(-c2ccccc2)c(-c2ncco2)cc1S(N)(=O)=O

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.47
EDNRB P24530 5/20 0.40
EDNRA P25101 5/20 0.40
CA1 P00915 4/20 0.40
CA2 P00918 4/20 0.40
CA12 O43570 3/20 0.40
CA9 Q16790 3/20 0.40
HPGDS O60760 1/20 0.40
HPGD P15428 2/20 0.39
CA4 P22748 1/20 0.38
CA7 P43166 1/20 0.38
BRD4 O60885 1/20 0.38
PIK3CD O00329 1/20 0.38
PIK3CG P48736 1/20 0.38
IMPDH2 P12268 1/20 0.38
LTA4H P09960 1/20 0.36
PDIA6 Q15084 1/20 0.35
ACLY P53396 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8554062 0.88 CA1 (0.44) MAOBEDNRBEDNRACA1CA2
SCHEMBL8551071 0.82 NTRK1 (0.41) MAOBEDNRBEDNRACA1CA2
SCHEMBL8547875 0.78 CA2 (0.45) MAOBCA1CA2CA12CA9
SCHEMBL7408121 0.78 HPGDS (0.44) MAOBEDNRBEDNRACA1CA2
SCHEMBL6026444 0.75 BRD4 (0.43) EDNRBEDNRACA1CA2CA12
SCHEMBL6986037 0.73 EDNRB (0.56) EDNRBEDNRAHPGDSLTA4H
SCHEMBL942521 0.73 HPGDS (0.47) MAOBEDNRBEDNRAHPGDSHPGD
SCHEMBL7408116 0.73 BRD4 (0.41) EDNRBEDNRACA1CA2CA12
SCHEMBL5174048 0.72 EDNRB (0.41) EDNRBEDNRAHPGDSHPGDBRD4
SCHEMBL19815373 0.70 HPGDS (0.45) HPGDSHPGDBRD4IMPDH2LTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5700816-A ANTIARTHRITIC AGENTS G.D. SEARLE & CO. 1997-12-23 US claimed
US-5700816-A ANTIARTHRITIC AGENTS G.D. SEARLE & CO. 1997-12-23 US disclosed