SCHEMBL8551071

SCHEMBL8551071

NS(=O)(=O)c1cc(-c2ncco2)c(-c2ccccc2)cc1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.41
CFTR P13569 1/20 0.39
CA2 P00918 7/20 0.39
CA1 P00915 6/20 0.39
CA12 O43570 3/20 0.39
CA9 Q16790 3/20 0.39
CA4 P22748 1/20 0.39
CA6 P23280 1/20 0.39
CA5A P35218 1/20 0.39
CA7 P43166 1/20 0.39
CA14 Q9ULX7 1/20 0.39
CA5B Q9Y2D0 1/20 0.39
S1PR1 P21453 2/20 0.38
S1PR3 Q99500 1/20 0.38
HPGDS O60760 1/20 0.37
SCN9A Q15858 1/20 0.35
NR1H2 P55055 1/20 0.35
NR1H3 Q13133 1/20 0.35
HPGD P15428 1/20 0.35
MAOB P27338 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8908949 0.85 ALOX5AP (0.40) CFTRCA2CA1CA12CA9
SCHEMBL8908994 0.82 MAOB (0.47) CA2CA1CA12CA9CA4
SCHEMBL8547875 0.75 CA2 (0.45) CA2CA1CA12CA9HPGDS
SCHEMBL6026444 0.72 BRD4 (0.43) CA2CA1CA12CA9CA4
SCHEMBL7408121 0.72 HPGDS (0.44) CA2CA1CA12CA9CA4
SCHEMBL6986037 0.71 EDNRB (0.56) HPGDSEDNRBEDNRA
SCHEMBL8554062 0.71 CA1 (0.44) CA2CA1CA12CA9CA4
SCHEMBL7408116 0.70 BRD4 (0.41) CA2CA1CA12CA9CA4
Trifluoroacetic Acid SCHEMBL27977019 0.68 PRSS1 (0.39) NTRK1CA2CA1CA12CA9
SCHEMBL5822874 0.68 PTGS2 (0.54) CA2CA1CA12CA9MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0825989-A1 SUBSTITUTED OXAZOLES FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1998-03-04 EP disclosed