SCHEMBL8909449

SCHEMBL8909449

COc1ccc(-c2oc(C(F)(F)F)nc2NS(=O)(=O)c2ccccc2)cc1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.42
PTGS1 P23219 4/20 0.41
HDAC6 Q9UBN7 3/20 0.41
HDAC4 P56524 2/20 0.41
HDAC1 Q13547 1/20 0.41
ERAP1 Q9NZ08 1/20 0.41
PPARA Q07869 1/20 0.40
PIK3CD O00329 1/20 0.40
SLC40A1 Q9NP59 1/20 0.40
MAPT P10636 2/20 0.39
LMNA P02545 2/20 0.39
TP53 P04637 1/20 0.39
HTR6 P50406 1/20 0.39
MIF P14174 1/20 0.39
POLB P06746 1/20 0.39
ABCB1 P08183 1/20 0.39
ABCC1 P33527 1/20 0.39
HSD11B1 P28845 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4405120 0.87 HDAC6 (0.45) HDAC6HDAC4HDAC1MAPTHSD11B1
SCHEMBL8560735 0.82 PTGS2 (0.43) PTGS2PTGS1PIK3CDSLC40A1MAPT
SCHEMBL8560251 0.81 HDAC6 (0.48) HDAC6HDAC4HDAC1MAPTLMNA
SCHEMBL8154450 0.80 KMO (0.47) HDAC6HDAC4HDAC1MAPTHSD11B1
Sulfamide SCHEMBL4639002 0.78 PTGS2 (0.46) PTGS2PTGS1MAPTMIFSMN1; SMN2
SCHEMBL9026371 0.78 KMT2A (0.41) PTGS2PTGS1PIK3CDSLC40A1MAPT
SCHEMBL8140595 0.77 MIF (0.43) PTGS2PTGS1MAPTMIFABCB1
SCHEMBL8631663 0.76 MAPK14 (0.46) PTGS2PTGS1ERAP1PPARAHTR6
SCHEMBL8629545 0.75 NPC1 (0.41) PTGS2PTGS1ERAP1PPARALMNA
SCHEMBL8153075 0.75 PTGS2 (0.55) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5700816-A ANTIARTHRITIC AGENTS G.D. SEARLE & CO. 1997-12-23 US claimed
US-5700816-A ANTIARTHRITIC AGENTS G.D. SEARLE & CO. 1997-12-23 US disclosed