SCHEMBL8909498

SCHEMBL8909498

CCOC(=O)C1=C(C)c2c(C)c3c(cc2=N1)-c1ccc(F)cc1N=3

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.37
GRM6 O15303 1/20 0.36
PRKCZ Q05513 1/20 0.36
CDC7 O00311 1/20 0.36
DBF4 Q9UBU7 1/20 0.36
MAPK14 Q16539 2/20 0.35
MAPT P10636 5/20 0.35
ALDH1A1 P00352 4/20 0.35
NPC1 O15118 3/20 0.35
RAB9A P51151 3/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
HPGD P15428 2/20 0.35
ALPL P05186 1/20 0.35
GAA P10253 1/20 0.35
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
CASP3 P42574 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
SENP7 Q9BQF6 1/20 0.34
TRPM8 Q7Z2W7 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8909809 0.91 TSHR (0.37) TSHRGRM6PRKCZMAPK14MAPT
SCHEMBL8910758 0.88 DHODH (0.38) TSHRMAPTALDH1A1NPC1RAB9A
SCHEMBL8909629 0.81 CA12 (0.39) MAPTALDH1A1SMN1; SMN2HPGDGAA
SCHEMBL9434374 0.80 SMAD3 (0.39) MAPTALDH1A1SMN1; SMN2GAANPSR1
SCHEMBL8909720 0.80 DHODH (0.38) MAPTALDH1A1NPC1RAB9AHPGD
SCHEMBL8912086 0.80 CYP2C9 (0.39) TSHRMAPTALDH1A1RAB9AHPGD
SCHEMBL8911562 0.80 POLB (0.40) GRM6PRKCZMAPTALDH1A1NPC1
SCHEMBL8910230 0.78 GABRA1 (0.38) TSHRMAPTALDH1A1SMN1; SMN2HPGD
SCHEMBL1388445 0.78 CA12 (0.37) MAPTALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL9434967 0.75 MAPT (0.42) TSHRMAPTALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5679694-A LOW TOXICITY AGAINST NORMAL CELL LINES THE WELLCOME FOUNDATION LTD. (GB) 1997-10-21 US disclosed
WO-1994002483-A1 TETRACYCLIC COMPOUNDS PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND THEIR USE AS ANTITUMOUR AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1994-02-03 WO disclosed