SCHEMBL8911562

SCHEMBL8911562

CCOC(=O)C1=C(C)c2c(C)c3c(cc2=N1)-c1cc(OC)ccc1N=3

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 4/20 0.38
KDM4E B2RXH2 3/20 0.38
ALDH1A1 P00352 3/20 0.38
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
MAPT P10636 2/20 0.38
PDE4D Q08499 1/20 0.38
PPARG P37231 5/20 0.38
CYP3A4 P08684 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.37
LMNA P02545 2/20 0.37
HTT P42858 1/20 0.37
PRKCZ Q05513 1/20 0.36
ATM Q13315 1/20 0.36
GABRG2 P18507 3/20 0.36
GABRB3 P28472 3/20 0.36
GABRA5 P31644 3/20 0.36
GRM6 O15303 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8909629 0.87 CA12 (0.39) GAAHPGDKDM4EALDH1A1MAPT
SCHEMBL9434374 0.86 SMAD3 (0.39) GAAALDH1A1MAPTHTTATM
SCHEMBL8912086 0.85 CYP2C9 (0.39) HPGDKDM4EALDH1A1RAB9AMAPT
SCHEMBL1388815 0.84 MAPT (0.44) GAAHPGDKDM4EALDH1A1NPC1
SCHEMBL8910230 0.83 GABRA1 (0.38) GAAHPGDKDM4EALDH1A1MAPT
SCHEMBL1388445 0.77 CA12 (0.37) POLBGAAHPGDKDM4EALDH1A1
SCHEMBL8910142 0.74 GAA (0.33) POLBGAAKDM4EALDH1A1NPC1
SCHEMBL9434967 0.74 MAPT (0.42) POLBGAAHPGDKDM4EALDH1A1
SCHEMBL8156114 0.73 CHRM2 (0.38) POLBGAAKDM4EALDH1A1MAPT
SCHEMBL8150571 0.72 HTT (0.32) ALDH1A1MAPTLMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5679694-A LOW TOXICITY AGAINST NORMAL CELL LINES THE WELLCOME FOUNDATION LTD. (GB) 1997-10-21 US claimed
EP-0651750-A1 TETRACYCLIC COMPOUNDS PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND THEIR USE AS ANTITUMOUR AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1995-05-10 EP disclosed
WO-1994002483-A1 TETRACYCLIC COMPOUNDS PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND THEIR USE AS ANTITUMOUR AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1994-02-03 WO disclosed