SCHEMBL8909543

SCHEMBL8909543

CC1=C(C(=O)n2ccnc2)N=c2cc3c(c(C)c21)=Nc1ccccc1-3

nearest known ligand 0.35

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
GPBAR1 Q8TDU6 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8142537 0.80 MYC (0.34) ALDH1A1
SCHEMBL8910392 0.80 CCNB2 (0.32) LMNA
SCHEMBL8536552 0.76 GAA (0.32) ALDH1A1LMNA
SCHEMBL9057850 0.75 MYC (0.36)
SCHEMBL8910714 0.74 ALDH1A1 (0.34) ALDH1A1LMNA
SCHEMBL8909578 0.74 HPGD (0.41) ALDH1A1
SCHEMBL8149445 0.72 TERT (0.36)
SCHEMBL8537456 0.72
SCHEMBL8154329 0.72 KMT2A (0.31) ALDH1A1LMNA
SCHEMBL8142555 0.71 NPC1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5679694-A LOW TOXICITY AGAINST NORMAL CELL LINES THE WELLCOME FOUNDATION LTD. (GB) 1997-10-21 US claimed
CN-1088209-A Heterogeneous ring compound WELLCOME FOUND (GB) 1994-06-22 CN disclosed
WO-1994002483-A1 TETRACYCLIC COMPOUNDS PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND THEIR USE AS ANTITUMOUR AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1994-02-03 WO disclosed