SCHEMBL8910392

SCHEMBL8910392

CC(=O)C1=C(C)c2c(C)c3c(cc2=N1)-c1ccccc1N=3

nearest known ligand 0.32

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCNB2 O95067 2/20 0.32
CDK1 P06493 2/20 0.32
CCNB1 P14635 2/20 0.32
GSK3A P49840 2/20 0.32
GSK3B P49841 2/20 0.32
CDK5 Q00535 2/20 0.32
CDK5R1 Q15078 2/20 0.32
CCNB3 Q8WWL7 2/20 0.32
MITF O75030 1/20 0.30
LMNA P02545 1/20 0.30
MAPT P10636 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8142537 0.90 MYC (0.34) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL8536552 0.85 GAA (0.32) LMNAMAPTHTT
SCHEMBL9057850 0.84 MYC (0.36)
SCHEMBL8909578 0.83 HPGD (0.41) MAPT
SCHEMBL8910714 0.83 ALDH1A1 (0.34) LMNAMAPTHTT
SCHEMBL8149445 0.81 TERT (0.36)
SCHEMBL8537456 0.81
SCHEMBL8154329 0.81 KMT2A (0.31) LMNAMAPT
SCHEMBL8148024 0.80 TDP2 (0.40) CCNB2CDK1CCNB1GSK3AGSK3B
SCHEMBL8909543 0.80 ALDH1A1 (0.33) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5679694-A LOW TOXICITY AGAINST NORMAL CELL LINES THE WELLCOME FOUNDATION LTD. (GB) 1997-10-21 US disclosed
WO-1994002483-A1 TETRACYCLIC COMPOUNDS PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND THEIR USE AS ANTITUMOUR AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1994-02-03 WO disclosed