SCHEMBL8910289

SCHEMBL8910289

CCCOP(=O)(Cc1nc(C2CCC2)cs1)OCCC

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.32
TMIGD3 P0DMS9 1/20 0.31
ADORA1 P30542 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8909261 0.90 RORC (0.33) RORCTMIGD3ADORA1
SCHEMBL9094297 0.68 TMIGD3 (0.36) RORCTMIGD3ADORA1
SCHEMBL22904608 0.67 MAPT (0.42) RORCTMIGD3ADORA1
SCHEMBL12790156 0.64 RORC (0.45) RORCTMIGD3ADORA1
SCHEMBL21417547 0.63 MAPT (0.34) RORC
SCHEMBL5708655 0.61 MAOA (0.47)
SCHEMBL24963463 0.61 MAPT (0.39) TMIGD3ADORA1
SCHEMBL18674653 0.61 ENPP2 (0.36) RORC
SCHEMBL21916139 0.60 CCNA2 (0.44)
SCHEMBL2227967 0.60 CTSK (0.38) RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5637720-A Intermediate for (E)-4-[[3-[2-(4-cycloalkyl-2-thiazolyl)ethenyl]phenyl]amino-2,2-alkyldiyl-4-oxobutanoic acids HOFFMANN-LA ROCHE INC. (US) 1997-06-10 US disclosed
WO-1996008479-A1 A PROCESS OF MAKING (E)-4-[3-[2-(4-CYCLOALKYL-2-THIAZOLYL)ETHENYL]PHENYL]AMINO-2,2-ALKYLDIYL-4-OXOBUTANOIC ACID F. HOFFMANN-LA ROCHE AG (CH) 1996-03-21 WO disclosed