SCHEMBL8910619

SCHEMBL8910619

[CH2]C(C)CS(=O)(=O)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PSIP1 O75475 1/20 0.56
HSD11B1 P28845 6/20 0.44
POLB P06746 1/20 0.43
ALDH1A1 P00352 3/20 0.42
TP53 P04637 1/20 0.42
HTT P42858 1/20 0.42
HSD17B10 Q99714 1/20 0.42
HTR6 P50406 1/20 0.41
CYP1A2 P05177 2/20 0.41
CYP2C19 P33261 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
GAA P10253 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
RCE1 Q9Y256 1/20 0.39
MMP1 P03956 1/20 0.39
MMP13 P45452 1/20 0.39
CYP2C9 P11712 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL778303 0.83 PSIP1 (0.60) PSIP1HSD11B1POLBALDH1A1TP53
SCHEMBL1972951 0.79 PSIP1 (0.56) PSIP1HSD11B1POLBALDH1A1TP53
SCHEMBL7724605 0.79 PSIP1 (0.56) PSIP1HSD11B1POLBALDH1A1TP53
SCHEMBL27596821 0.79 PSIP1 (0.56) PSIP1HSD11B1POLBALDH1A1TP53
SCHEMBL8909374 0.79 PSIP1 (0.56) PSIP1HSD11B1POLBALDH1A1TP53
SCHEMBL9426107 0.79 PSIP1 (0.56) PSIP1HSD11B1POLBALDH1A1TP53
SCHEMBL6181714 0.79 PSIP1 (0.50) PSIP1HSD11B1POLBALDH1A1TP53
SCHEMBL17018545 0.78 PSIP1 (0.54) PSIP1HSD11B1POLBALDH1A1SMN1; SMN2
SCHEMBL2444476 0.78 PSIP1 (0.59) PSIP1HSD11B1POLBALDH1A1TP53
SCHEMBL7347205 0.78 PSIP1 (0.54) PSIP1HSD11B1POLBALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0813543-A1 BIS-AMINO ACID HYDROXYETHYLAMINO SULFONAMIDE RETROVIRAL PROTEASE INHIBITORS G.D. SEARLE & CO. (US) 1997-12-29 EP disclosed
WO-1996028464-A1 BIS-AMINO ACID HYDROXYETHYLAMINO SULFONAMIDE RETROVIRAL PROTEASE INHIBITORS G.D. SEARLE & CO. (US) 1996-09-19 WO disclosed
CN-1114834-A antidiabetic agent OTSUKA PHARMA CO LTD (JP) 1996-01-10 CN disclosed
EP-0670831-A1 QUINOXALINE DERIVATIVE AS ANTIDIABETIC AGENT OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-09-13 EP disclosed
WO-1995009159-A1 QUINOXALINE DERIVATIVE AS ANTIDIABETIC AGENT OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1995-04-06 WO disclosed