SCHEMBL8910680

SCHEMBL8910680

NC(=O)c1cccc(-c2cccc3ccccc23)c1C(N)=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.51
GAA P10253 2/20 0.51
ALDH1A1 P00352 2/20 0.51
POLB P06746 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
NR4A1 P22736 1/20 0.48
NR4A2 P43354 1/20 0.48
NR4A3 Q92570 1/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
BCAT2 O15382 1/20 0.47
ALOX5 P09917 1/20 0.47
KEAP1 Q14145 1/20 0.46
NFE2L2 Q16236 1/20 0.46
RORC P51449 1/20 0.44
RORB Q92753 1/20 0.44
MMP3 P08254 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
PTPN1 P18031 1/20 0.43
CDC25B P30305 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31154022 0.90 NR4A1 (0.59) KDM4EGAAALDH1A1POLBSMN1; SMN2
SCHEMBL209369 0.90 NR4A1 (0.59) KDM4EGAAALDH1A1POLBSMN1; SMN2
SCHEMBL27830752 0.90 NR4A1 (0.55) KDM4EGAAALDH1A1POLBSMN1; SMN2
SCHEMBL30892682 0.89 BCAT2 (0.55) KDM4EGAAALDH1A1POLBSMN1; SMN2
SCHEMBL5849850 0.89 BCAT2 (0.55) KDM4EGAAALDH1A1POLBSMN1; SMN2
SCHEMBL31621277 0.89 BCAT2 (0.55) KDM4EGAAALDH1A1POLBSMN1; SMN2
SCHEMBL402013 0.84 BCAT2 (0.56) KDM4EGAAALDH1A1BCAT2KEAP1
SCHEMBL28323302 0.84 KDM4E (0.50) KDM4EGAAALDH1A1POLBSMN1; SMN2
SCHEMBL9068297 0.84 KEAP1 (0.56) KDM4EGAAALDH1A1POLBSMN1; SMN2
SCHEMBL28053358 0.83 KDM4E (0.49) KDM4EGAAALDH1A1POLBSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0804643-A2 WATER CONTAINING AROMATIC POLYAMIDE PULP AND PROCESS FOR PRODUCING THE SAME Akzo Nobel N.V. (NL) 1997-11-05 EP disclosed
EP-0741813-A1 AROMATIC POLYAMIDE PULP AND ITS PRODUCTION PROCESS Akzo Nobel N.V. (NL) 1996-11-13 EP disclosed
WO-1995030044-A2 WATER CONTAINING AROMATIC POLYAMIDE PULP AND PROCESS FOR PRODUCING THE SAME AKZO NOBEL N.V. (NL) 1995-11-09 WO disclosed
WO-1995019466-A1 AROMATIC POLYAMIDE PULP AND ITS PRODUCTION PROCESS AKZO NOBEL N.V. (NL) 1995-07-20 WO disclosed
EP-0658226-A1 WATER-CONTAINING AROMATIC POLYAMIDE PULP AND PROCESS FOR PRODUCING THE SAME. AKZO NOBEL NV (NL) 1995-06-21 EP disclosed
WO-1994005854-A1 WATER-CONTAINING AROMATIC POLYAMIDE PULP AND PROCESS FOR PRODUCING THE SAME AKZO NOBEL N.V. (NL) 1994-03-17 WO disclosed
US-4868041-A AROMATIC POLYAMIDES, COMPOSITES YARNS, CORES TOYO BOSEKI KABUSHIKI KAISHA (JP) 1989-09-19 US disclosed