SCHEMBL8910992

SCHEMBL8910992

O=[C]C1c2ccccc2CC(=O)c2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.44
BCHE P06276 1/20 0.44
KDM4E B2RXH2 3/20 0.42
ALDH1A1 P00352 3/20 0.42
HPGD P15428 2/20 0.42
ANPEP P15144 2/20 0.41
MAOA P21397 2/20 0.38
HTR2A P28223 3/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
PABPC1 P11940 1/20 0.36
BLM P54132 1/20 0.36
CYP2A6 P11509 1/20 0.35
MAOB P27338 1/20 0.35
HRH1 P35367 2/20 0.34
HTR2C P28335 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL68229 0.77 GPR3 (0.41) ALDH1A1HTR2AMEN1KMT2AHDAC4
SCHEMBL9187132 0.75 ACP3 (0.48) CES1HTR2A
SCHEMBL22879435 0.75 BCHE (0.47) CES1BCHEKDM4EALDH1A1HPGD
SCHEMBL21312228 0.75 CES1 (0.47) CES1BCHEKDM4EALDH1A1HPGD
SCHEMBL24119326 0.71 BCHE (0.43) CES1BCHEKDM4EALDH1A1HPGD
SCHEMBL8035811 0.70 CES1 (0.73) CES1BCHEKDM4EALDH1A1HPGD
SCHEMBL569873 0.70
SCHEMBL31070117 0.70
SCHEMBL8506762 0.68 ALDH1A1 (0.41) CES1BCHEKDM4EALDH1A1HPGD
SCHEMBL2680028 0.67 S100A4 (0.41) CES1BCHEKDM4EALDH1A1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5622953-A DRUG RESISTANT TO ANTICANCER CHEMOTHERAPEUTIC DRUG BASF AKTIENGESELLSCHAFT (DE) 1997-04-22 US disclosed
EP-0691962-A1 1-AMINO-3-PHENOXY PROPANE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE BASF AKTIENGESELLSCHAFT (DE) 1996-01-17 EP disclosed
WO-1994022842-A1 1-AMINO-3-PHENOXY PROPANE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE BASF AKTIENGESELLSCHAFT (DE) 1994-10-13 WO disclosed