SCHEMBL8911202

SCHEMBL8911202

[c]1ccc2c(c1)CNCc1ccccc1-2

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.38
CA9 Q16790 1/20 0.38
MAOB P27338 2/20 0.36
PNMT P11086 1/20 0.36
CD44 P16070 1/20 0.36
OXTR P30559 1/20 0.33
PRCP P42785 1/20 0.32
RYR2 Q92736 1/20 0.32
MAOA P21397 1/20 0.31
HTR2C P28335 1/20 0.31
METAP2 P50579 1/20 0.31
MEN1 O00255 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
KMT2A Q03164 1/20 0.30
PARP1 P09874 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1165406 0.81 CA12 (0.52) CA12CA9MAOBPNMTCD44
Hydrochloric Acid SCHEMBL32672905 0.79 CA12 (0.50) CA12CA9MAOBPNMTCD44
SCHEMBL24657 0.78 MAOA (0.46) MAOBPNMTMAOAHTR2CMETAP2
SCHEMBL476341 0.78 CES1 (0.46) MAOBMAOAPARP1
Water SCHEMBL28256098 0.71 PNMT (0.62) MAOBPNMTCD44OXTRPRCP
SCHEMBL24206 0.69 MAOA (0.46) MAOBPNMTMAOAHTR2CMETAP2
SCHEMBL4312831 0.69 CES1 (0.46) MAOBMAOAPARP1
SCHEMBL71211 0.69
SCHEMBL134194 0.69
SCHEMBL6293496 0.69 CA12 (0.38) CA12CA9MAOBPNMTCD44

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5686466-A CHOLINESERASE INHIBITOR; TREATMENT OF SENILE DEMENTIA, ALZHEIMER'S DISEASE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-11-11 US claimed
EP-0607864-A2 Tricyclic condensed heterocyclic compounds for the treatment of senile dementic Takeda Chemical Industries, Ltd. (JP) 1994-07-27 EP claimed