SCHEMBL8910142

SCHEMBL8910142

CCOC(=O)C1=C(C)c2c(C)c3c(cc2=N1)-c1ccc(OC(C)=O)c(OC)c1N=3

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.33
MAPT P10636 3/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
HSD17B10 Q99714 1/20 0.32
SLC10A2 Q12908 1/20 0.32
PTPN1 P18031 2/20 0.31
POLB P06746 1/20 0.31
LMNA P02545 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
TNFSF11 O14788 1/20 0.30
ABCG2 Q9UNQ0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1388445 0.79 CA12 (0.37) GAAMAPTALDH1A1KDM4ENPC1
SCHEMBL8911562 0.74 POLB (0.40) GAAMAPTALDH1A1KDM4ENPC1
SCHEMBL8909629 0.72 CA12 (0.39) GAAMAPTALDH1A1KDM4EHSD17B10
SCHEMBL8911173 0.69 TDP1 (0.39) MAPTALDH1A1NPC1RAB9APOLB
SCHEMBL9435019 0.66 ALDH1A1 (0.35) GAAMAPTALDH1A1KDM4ENPC1
SCHEMBL7965437 0.66 KDM4E (0.34) GAAMAPTALDH1A1KDM4ENPC1
SCHEMBL9434967 0.64 MAPT (0.42) GAAMAPTALDH1A1KDM4ENPC1
SCHEMBL8150571 0.62 HTT (0.32) MAPTALDH1A1LMNASMN1; SMN2
SCHEMBL28659592 0.60 TSHR (0.50) GAAMAPTALDH1A1KDM4ENPC1
SCHEMBL4647233 0.60 HSD17B2 (0.66) GAAMAPTALDH1A1KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5679694-A LOW TOXICITY AGAINST NORMAL CELL LINES THE WELLCOME FOUNDATION LTD. (GB) 1997-10-21 US disclosed
EP-0651750-A1 TETRACYCLIC COMPOUNDS PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND THEIR USE AS ANTITUMOUR AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1995-05-10 EP disclosed
WO-1994002483-A1 TETRACYCLIC COMPOUNDS PROCESS AND INTERMEDIATES FOR THEIR PREPARATION AND THEIR USE AS ANTITUMOUR AGENTS THE WELLCOME FOUNDATION LIMITED (GB) 1994-02-03 WO disclosed