Levofloxacin Anhydrous

Levofloxacin Anhydrous

SCHEMBL891190

C[C@H]1COc2c(N3CCN(C)CC3)c(F)cc3c(=O)c(C(=O)O)cn1c23.O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

gyrAgyrBparCparE

The experimentally established mechanism targets of Levofloxacin Anhydrous. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 1.00
TUBB4A P04350 7/20 1.00
TUBB P07437 7/20 1.00
TUBA3C P0DPH7 7/20 1.00
TUBA1B P68363 7/20 1.00
TUBA4A P68366 7/20 1.00
TUBB4B P68371 7/20 1.00
TUBB3 Q13509 7/20 1.00
TUBB2A Q13885 7/20 1.00
TUBB8 Q3ZCM7 7/20 1.00
TUBA3E Q6PEY2 7/20 1.00
TUBA1A Q71U36 7/20 1.00
TUBA1C Q9BQE3 7/20 1.00
TUBB6 Q9BUF5 7/20 1.00
TUBB2B Q9BVA1 7/20 1.00
TUBB1 Q9H4B7 7/20 1.00
POLB P06746 1/20 1.00
SLC47A1 Q96FL8 1/20 1.00
RCE1 Q9Y256 1/20 1.00
ALDH1A1 P00352 5/20 0.98

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ofloxacin SCHEMBL6090650 1.00 KDM4E (1.00) KDM4ETUBB4ATUBBTUBA3CTUBA1B
Ofloxacin SCHEMBL6092282 1.00 KDM4E (1.00) KDM4ETUBB4ATUBBTUBA3CTUBA1B
Levofloxacin Anhydrous SCHEMBL1650602 1.00 KDM4E (1.00) KDM4ETUBB4ATUBBTUBA3CTUBA1B
Levofloxacin Anhydrous SCHEMBL30009030 1.00 KDM4E (1.00) KDM4ETUBB4ATUBBTUBA3CTUBA1B
Levofloxacin Anhydrous SCHEMBL27810870 0.99 KDM4E (0.98) KDM4ETUBB4ATUBBTUBA3CTUBA1B
Ofloxacin SCHEMBL9745243 0.99 KDM4E (1.00) KDM4ETUBB4ATUBBTUBA3CTUBA1B
Dextrofloxacine SCHEMBL4316947 0.99 KDM4E (1.00) KDM4ETUBB4ATUBBTUBA3CTUBA1B
Ofloxacin SCHEMBL14163982 0.99 KDM4E (1.00) KDM4ETUBB4ATUBBTUBA3CTUBA1B
Ofloxacin SCHEMBL5532921 0.99 KDM4E (1.00) KDM4ETUBB4ATUBBTUBA3CTUBA1B
Ofloxacin SCHEMBL24373 0.99 KDM4E (1.00) KDM4ETUBB4ATUBBTUBA3CTUBA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 171 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119562814-A Otologic liquid for preventing and/or treating otitis externa and/or otitis media 西奥利亚制药株式会社 2025-03-04 CN claimed
WO-2023224045-A1 OTOLOGICAL SOLUTION FOR PREVENTING AND/OR TREATING OTITIS EXTERNA AND/OR OTITIS MEDIA セオリアファーマ株式会社 2023-11-23 WO claimed
CN-108310983-B Preparation and regeneration method of antibacterial and anti-pollution PVDF ultrafiltration membrane 山西大学 2021-02-02 CN claimed
US-9603805-B2 Easily dosable solid preparation MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 2017-03-28 US claimed
CN-103813807-B Easily administrable solid preparation 持田制药株式会社 2017-02-08 CN claimed
US-20140308359-A1 EASILY DOSABLE SOLID PREPARATION MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 2014-10-16 US claimed
EP-2762167-A1 EASY-TO-TAKE SOLID PREPARATION Mochida Pharmaceutical Co., Ltd. (JP) 2014-08-06 EP claimed
US-7678903-B2 Preparation of levofloxacin hemihydrate free of levofloxacin monohydrate by reacting (S)-(-) 9,10-difluoro-3-methyl-7-oxo-2,3-dihydro-7H-pyrido[1,2,3-de][1,4] benzoxazine-6-carboxylic acid with N-methyl piperazine to yield crude levofloxacin which is suspended in isopropanol, adding water, precipitating MATRIX LABORATORIES LIMITED (IN) 2010-03-16 US claimed
US-7629458-B2 Preparation of levofloxacin and hemihydrate thereof TEVA PHARMACEUTICAL INDUSTRIES LTD. (IL) 2009-12-08 US claimed
US-20080097095-A1 Process for the Preparation of Levofloxacin Hemiydrate MYLAN LABORATORIES LIMITED (IN) 2008-04-24 US claimed
US-20060276463-A1 Pure levofloxacin hemihydrate and processes for preparation thereof RANBAXY LABORATORIES LIMITED (IN) 2006-12-07 US claimed
CN-1735620-A Pure levofloxacin hemihydrate and process for its preparation RANBAXY LAB LTD (IN) 2006-02-15 CN claimed
WO-2004055025-A1 PURE LEVOFLOXACIN HEMIHYDRATE AND PROCESSES FOR PREPARATION THEREOF RANBAXY LABORATORIES LIMITED (IN) 2004-07-01 WO claimed
EP-0444678-B1 Process for selectively producing hydrate crystals DAIICHI SEIYAKU CO (JP) 1997-09-03 EP claimed
US-5545737-A Process for selectively producing an (S)-9-fluoro-3-methyl-10-(4-methyl-1-piperazinyl)-7-oxo-2,3-dihydro-7h-pyrido (1,2,3, -de) (1,4) benzoxazine-6-carboxylic acid hemihydrate or monohydrate DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1996-08-13 US claimed
EP-0444678-A1 Process for selectively producing hydrate crystals DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1991-09-04 EP claimed
EP-4039257-B1 PHARMACEUTICAL COMPOSITION AND KIT CONTAINING A PENAM DERIVATIVE OR SALT THEREOF AND ONE OR MORE COMPOUNDS SELECTED FROM BETA-LACTAMASE INHIBITOR COMPOUND, ANTIBACTERIAL COMPOUND AND SALTS OF THESE FUJIFILM CORP (JP) 2026-05-27 EP disclosed
US-20260091082-A1 CYCLIC PEPTIDE DERIVATIVE COMPOSITION FOR TREATING OR PREVENTING EYE DISEASE DKS CO. LTD. (JP) 2026-04-02 US disclosed
US-5023257-A Related to ciprofloxacin, in the form of oily suspension; bacterial infections BAYER AKTIENGESELLSCHAFT (DE) 1991-06-11 US disclosed
EP-0394553-A2 Use of fluorine containing pyridone carboxylic acid derivatives for preparing a medicament for the treatment of HIV infections DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1990-10-31 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060276463-A1 Pure levofloxacin hemihydrate and processes for preparation thereof CYP4F3, QARS1, CYP4F11 KDM4E 942/4885TUBB4A 1662/4885TUBB 1745/4885
US-20260091082-A1 CYCLIC PEPTIDE DERIVATIVE COMPOSITION FOR TREATING OR PREVENTING EYE DISEASE ADCY3, GLP1R, PDE6C KDM4E 4379/4885TUBB4A 4786/4885TUBB 4710/4885
US-20080097095-A1 Process for the Preparation of Levofloxacin Hemiydrate CYP4F3, HPD, CYP4F11 KDM4E 645/4885TUBB4A 2364/4885TUBB 2337/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.