SCHEMBL8912045

SCHEMBL8912045

Cc1c(NC(=O)c2ccccc2)sc2nc(C(N)CC(=O)OCc3ccccc3)oc(=O)c12

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 3/20 0.43
MAPT P10636 3/20 0.43
HPGD P15428 3/20 0.43
NPSR1 Q6W5P4 1/20 0.39
ADORA3 P0DMS8 1/20 0.39
ADORA2A P29274 1/20 0.39
ELANE P08246 1/20 0.37
MEN1 O00255 1/20 0.37
POLB P06746 1/20 0.37
GAA P10253 1/20 0.37
KMT2A Q03164 1/20 0.37
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8911361 0.90 NPSR1 (0.39) ALDH1A1HPGDNPSR1ELANETSHR
SCHEMBL8912018 0.90 ALDH1A1 (0.39) ALDH1A1MAPTNPSR1ELANEMEN1
SCHEMBL8911896 0.89 ATM (0.38) ALDH1A1NPSR1ELANESMN1; SMN2
SCHEMBL8913772 0.89 ITGB3 (0.39) ALDH1A1NPSR1
SCHEMBL8911768 0.87 ALDH1A1 (0.39) ALDH1A1KDM4EMAPTNPSR1MEN1
SCHEMBL8917887 0.86 MAPT (0.40) ALDH1A1KDM4EMAPTHPGDNPSR1
SCHEMBL8913843 0.86 NPSR1 (0.36) ALDH1A1NPSR1ELANETSHRSMN1; SMN2
SCHEMBL8913653 0.85 ALDH1A1 (0.41) ALDH1A1ELANETSHRSMN1; SMN2
SCHEMBL8912049 0.85 ATM (0.53) NPSR1
SCHEMBL8911749 0.84 ALDH1A1 (0.41) ALDH1A1ELANETSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799230-A1 THIENOXAZINONE DERIVATIVES USEFUL AS ANTIVIRAL AGENTS SMITHKLINE BEECHAM PLC (GB) 1997-10-08 EP disclosed
WO-1996019482-A1 THIENOXAZINONE DERIVATIVES USEFUL AS ANTIVIRAL AGENTS SMITHKLINE BEECHAM PLC (GB) 1996-06-27 WO disclosed