SCHEMBL8912082

SCHEMBL8912082

CCCCCC(O)c1nccn1C(c1ccccc1)(c1ccccc1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.38
KMT2A Q03164 3/20 0.35
MEN1 O00255 1/20 0.35
CSNK1E P49674 1/20 0.35
HSP90AA1 P07900 1/20 0.35
CYP2D6 P10635 1/20 0.34
LMNA P02545 1/20 0.34
KCNA5 P22460 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5692289 0.86 KDM4E (0.41) KDM4EKMT2AMEN1CYP2D6LMNA
SCHEMBL9238656 0.79 KDM4E (0.44) KDM4EKMT2AMEN1CYP2D6
SCHEMBL6321358 0.78 KDM4E (0.37) KDM4EKMT2AMEN1CYP2D6
SCHEMBL9628706 0.75 LMNA (0.56) KMT2ACYP2D6LMNA
SCHEMBL8806973 0.73 KMT2A (0.42) KMT2AMEN1KCNH2
SCHEMBL20768154 0.72 KMT2A (0.38) KDM4EKMT2AMEN1CYP2D6
SCHEMBL28203075 0.72 MAPT (0.47) KMT2A
SCHEMBL18007731 0.71 KMT2A (0.35) KMT2AMEN1HSP90AA1
SCHEMBL28942503 0.71 L3MBTL1 (0.46) KDM4EKMT2ACYP2D6LMNA
SCHEMBL28202269 0.71 TLR8 (0.37) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5693633-A Angiotensin II antagonists ELI LILLY AND COMPANY (US) 1997-12-02 US disclosed
US-5612360-A AROMATIC N-HETEROCYCLIC COMPOUNDS AS HYPOTENSIVE AGENTS WITH ACID GROUPS, SULFONYLCARBOXAMIDES OR TETRAZOLE GROUPS ELI LILLY AND COMPANY (US) 1997-03-18 US disclosed
US-5569768-A USEFUL IN TREATING HYPERTENSION, CONGESTIVE HEART FAILURE, GLAUCOMA AND RENAL INSUFFICIENCY ELI LILLY AND COMPANY (US) 1996-10-29 US disclosed
US-5556981-A Angiotensin II antagonist intermediates ELI LILLY AND COMPANY (US) 1996-09-17 US disclosed
CN-1101908-A Angiotensin II antagonists LILLY CO ELI (US) 1995-04-26 CN disclosed
EP-0574174-A2 Angiotensin II antagonists ELI LILLY AND COMPANY (US) 1993-12-15 EP disclosed