SCHEMBL8912487

SCHEMBL8912487

CS(=O)(=O)Nc1ccc2c(c1)C(=O)C1(CCNCC1)C2

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 3/20 0.42
PDPK1 O15530 3/20 0.40
MET P08581 1/20 0.39
KDM1A O60341 3/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
ALDH1A1 P00352 1/20 0.37
AURKA O14965 1/20 0.36
KDR P35968 1/20 0.36
AURKB Q96GD4 1/20 0.36
KAT2B Q92831 1/20 0.36
HTR6 P50406 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30341566 1.00 TDP2 (0.42) TDP2PDPK1METKDM1AMAOA
SCHEMBL8915989 0.88 MET (0.43) TDP2PDPK1METKDM1AMAOA
Hydrochloric Acid SCHEMBL8912504 0.87 MET (0.42) TDP2PDPK1METKDM1AMAOA
SCHEMBL22770286 0.79 MET (0.38) TDP2METKDM1A
SCHEMBL8914677 0.79 SMN1; SMN2 (0.44) TDP2KDM1AALDH1A1
SCHEMBL21856169 0.77 F7 (0.44) TDP2
SCHEMBL29506005 0.77 F7 (0.44) TDP2
SCHEMBL8914076 0.76 KCNH2 (0.51)
SCHEMBL28905294 0.75 PARP10 (0.44) TDP2KDRAURKB
SCHEMBL28464048 0.75 PARP1 (0.44) TDP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP disclosed