SCHEMBL8915989

SCHEMBL8915989

CS(=O)(=O)Nc1ccc2c(c1)C(=O)C1(CCNCC1)CC2

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MET P08581 1/20 0.43
TDP2 O95551 3/20 0.41
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38
HTR2B P41595 2/20 0.38
SIGMAR1 Q99720 2/20 0.38
KDM1A O60341 2/20 0.38
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
HTR6 P50406 1/20 0.38
NR3C1 P04150 1/20 0.38
PGR P06401 1/20 0.38
NR3C2 P08235 1/20 0.38
AR P10275 1/20 0.38
PDPK1 O15530 3/20 0.37
HTR1A P08908 1/20 0.37
HTR7 P34969 1/20 0.37
ALDH1A1 P00352 1/20 0.36
AURKA O14965 1/20 0.36
KDR P35968 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8912504 0.99 MET (0.42) METTDP2HTR2AHTR2CHTR2B
SCHEMBL30341566 0.88 TDP2 (0.42) METTDP2KDM1AMAOAMAOB
SCHEMBL8912487 0.88 TDP2 (0.42) METTDP2KDM1AMAOAMAOB
SCHEMBL8913831 0.80 HTR2A (0.42) METHTR2AHTR2CHTR2BSIGMAR1
SCHEMBL8913620 0.76 SIGMAR1 (0.56) HTR2AHTR2CHTR2BSIGMAR1
SCHEMBL8568665 0.72 PKM (0.44) HTR2AHTR6NR3C2
SCHEMBL10360424 0.71 HTR6 (0.66) HTR2AHTR2CHTR2BHTR6ALDH1A1
SCHEMBL1912704 0.71 SIGMAR1 (0.64) HTR2AHTR2CHTR2BSIGMAR1MAOA
SCHEMBL6841697 0.71 ADRA2A (0.47) TDP2HTR2AHTR2CHTR2BSIGMAR1
Hydrochloric Acid SCHEMBL8565340 0.71 PKM (0.43) HTR6NR3C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP disclosed