SCHEMBL8913591

SCHEMBL8913591

CC(=O)N1CCC2(CC1)Cc1ccc(N)cc1C2=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GFER P55789 2/20 0.41
CASP6 P55212 1/20 0.41
USP2 O75604 2/20 0.36
HSD17B10 Q99714 3/20 0.36
CASP1 P29466 2/20 0.36
CASP7 P55210 2/20 0.36
ALDH1A1 P00352 4/20 0.35
CYP2C19 P33261 2/20 0.35
MAPK1 P28482 2/20 0.35
CYP3A4 P08684 2/20 0.35
HIF1A Q16665 1/20 0.35
HSD17B3 P37058 1/20 0.35
KDM4E B2RXH2 2/20 0.35
HPGD P15428 2/20 0.35
BAZ2B Q9UIF8 1/20 0.35
BACE1 P56817 1/20 0.35
AKT1 P31749 1/20 0.35
CYP2C9 P11712 3/20 0.35
TSHR P16473 1/20 0.35
GAA P10253 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8913172 0.88 SIGMAR1 (0.47) GFERCASP6HSD17B10CASP1CASP7
SCHEMBL22770382 0.88 ALDH1A1 (0.36) HSD17B10CASP1CASP7ALDH1A1KDM4E
SCHEMBL29993019 0.83 NR1H2 (0.53) ALDH1A1MAPK1NR1H2
SCHEMBL22770482 0.83 NR1H2 (0.53) ALDH1A1MAPK1NR1H2
SCHEMBL8916017 0.81 HTR2A (0.52) GFERUSP2HSD17B10ALDH1A1CYP2C19
SCHEMBL8913519 0.80 ALDH1A1 (0.45) ALDH1A1HPGDBAZ2BGAAKMT2A
SCHEMBL8914677 0.79 SMN1; SMN2 (0.44) ALDH1A1GAASMN1; SMN2
SCHEMBL31288591 0.73 OTUD7B (0.42) ALDH1A1CYP2C19CYP3A4KDM4EHPGD
SCHEMBL20511922 0.72 CA1 (0.36) ALDH1A1CYP2C19CYP2C9KMT2ASMN1; SMN2
SCHEMBL22770466 0.70 OTUD7B (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP disclosed