SCHEMBL8913639

SCHEMBL8913639

CC(=O)N1CCC2(CC1)Cc1cc(NS(C)(=O)=O)ccc1O2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 3/20 0.46
HDAC3 O15379 2/20 0.45
HDAC4 P56524 2/20 0.45
HDAC1 Q13547 2/20 0.45
HDAC7 Q8WUI4 2/20 0.45
HDAC2 Q92769 2/20 0.45
HDAC10 Q969S8 2/20 0.45
HDAC11 Q96DB2 2/20 0.45
HDAC8 Q9BY41 2/20 0.45
HDAC6 Q9UBN7 2/20 0.45
HDAC9 Q9UKV0 2/20 0.45
HDAC5 Q9UQL6 2/20 0.45
KCNH2 Q12809 1/20 0.44
KDM4E B2RXH2 2/20 0.44
ALDH1A1 P00352 2/20 0.44
GAA P10253 2/20 0.44
KMT2A Q03164 2/20 0.44
MEN1 O00255 1/20 0.44
MAPT P10636 1/20 0.44
ADRA1A P35348 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8912969 0.87 HDAC3 (0.48) ADRA1DHDAC3HDAC4HDAC1HDAC7
SCHEMBL8913770 0.80 ADRA1D (0.41) ADRA1DKCNH2ADRA1AADRA1B
SCHEMBL8569459 0.78 EPHX2 (0.56) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL8564005 0.76 ADRA1D (0.66) ADRA1DHDAC3HDAC4HDAC1HDAC7
SCHEMBL11257265 0.75 TRPM8 (0.52) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL8912479 0.74 ALDH1A1 (0.45) HDAC3HDAC4HDAC1HDAC7HDAC2
SCHEMBL262004 0.74 HDAC3 (0.66) ADRA1DHDAC3HDAC4HDAC1HDAC7
SCHEMBL8914677 0.74 SMN1; SMN2 (0.44) ADRA1DALDH1A1GAAADRA1AADRA1B
SCHEMBL8914795 0.74 HDAC3 (0.41) ADRA1DHDAC3HDAC4HDAC1HDAC7
Hydrochloric Acid SCHEMBL8912935 0.73 HDAC3 (0.41) ADRA1DHDAC3HDAC4HDAC1HDAC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5633247-A ANTIARRTHYMIA AGENT MERCK & CO., INC. (US) 1997-05-27 US disclosed
US-5206240-A Antiarrhythmia agents MERCK & CO., INC. (US) 1993-04-27 US disclosed
EP-0431943-A2 Nitrogen-containing spirocycles MERCK & CO. INC. (US) 1991-06-12 EP disclosed