SCHEMBL8914486

SCHEMBL8914486

Cc1c(SCCN2CCOCC2)ccnc1CSc1nc2ccccc2n1CCO

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.49
HPGD P15428 2/20 0.49
LMNA P02545 2/20 0.47
ALDH1A1 P00352 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2C19 P33261 2/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
PDE10A Q9Y233 1/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
MAPT P10636 2/20 0.42
TP53 P04637 1/20 0.42
HSD17B10 Q99714 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
CASP1 P29466 1/20 0.42
CASP7 P55210 1/20 0.42
RAB9A P51151 1/20 0.40
MAPK1 P28482 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5109272 0.89 CYP3A4 (0.52) ALDH1A1CYP3A4CYP2C19MAPTTP53
SCHEMBL8916260 0.87 MAPT (0.54) KDM4EHPGDALDH1A1CYP3A4CYP2C19
SCHEMBL8915650 0.87 CYP3A4 (0.48) KDM4EHPGDLMNAALDH1A1CYP3A4
SCHEMBL8914024 0.83 L3MBTL1 (0.45) KDM4EHPGDALDH1A1PDE10AMAPT
SCHEMBL8914183 0.83 GAA (0.50) KDM4EHPGDALDH1A1PDE10AMEN1
SCHEMBL5106665 0.82 PDE10A (0.43) KDM4EHPGDLMNAALDH1A1CYP3A4
SCHEMBL5120357 0.81 PDE10A (0.42) KDM4ELMNAALDH1A1CYP3A4CYP2C19
SCHEMBL8916044 0.77 USP2 (0.49) KDM4EHPGDLMNAALDH1A1PDE10A
SCHEMBL8915606 0.77 RAB9A (0.69) HPGDALDH1A1CYP3A4CYP2C19CYP1A2
SCHEMBL8915212 0.77 KDM4E (0.43) KDM4EHPGDLMNAALDH1A1PDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5616581-A BACTERICIDES YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-04-01 US disclosed
US-5504082-A BACTERICIDE FOR HELICOBACTER, ANTIULCER AGENT, GASTRIC ACIDSUPPRESSOR YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-04-02 US disclosed
EP-0644191-A1 PYRIDINE COMPOUND AND MEDICINAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1995-03-22 EP disclosed