SCHEMBL8914889

SCHEMBL8914889

Cc1c(SCCN2CCc3ccccc3C2)ccnc1CSc1nc2ncccc2[nH]1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 2/20 0.47
RAB9A P51151 5/20 0.44
SMN1; SMN2 Q16637 4/20 0.44
NPC1 O15118 4/20 0.44
HPGD P15428 4/20 0.44
TP53 P04637 5/20 0.44
PDE10A Q9Y233 1/20 0.42
ALDH1A1 P00352 3/20 0.41
BACE1 P56817 1/20 0.41
HSD17B10 Q99714 1/20 0.41
THRB P10828 2/20 0.41
KDM4E B2RXH2 1/20 0.41
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
POLB P06746 1/20 0.40
RXFP1 Q9HBX9 1/20 0.39
DRD2 P14416 2/20 0.38
DRD3 P35462 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8914916 0.90 RAB9A (0.49) GRIN2BRAB9ANPC1PDE10AALDH1A1
SCHEMBL8914888 0.86 DRD2 (0.42) RAB9ANPC1ALDH1A1HSD17B10KDM4E
SCHEMBL8915115 0.85 RAB9A (0.40) GRIN2BRAB9ASMN1; SMN2NPC1ALDH1A1
SCHEMBL8915109 0.85 RAB9A (0.43) RAB9ASMN1; SMN2NPC1HPGDTP53
SCHEMBL7849078 0.79 TP53 (0.41) GRIN2BRAB9ASMN1; SMN2NPC1HPGD
SCHEMBL8805150 0.78 RAB9A (0.54) GRIN2BRAB9ASMN1; SMN2NPC1HPGD
SCHEMBL8914425 0.78 ALDH1A1 (0.52) ALDH1A1KDM4EDRD2DRD3LMNA
SCHEMBL8915296 0.78 KDM4E (0.52) ALDH1A1KDM4EPOLBDRD2DRD3
Hydrochloric Acid SCHEMBL8430958 0.77 RAB9A (0.53) GRIN2BRAB9ASMN1; SMN2NPC1HPGD
SCHEMBL8915325 0.76 RAB9A (0.55) GRIN2BRAB9ASMN1; SMN2NPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0644191-A1 PYRIDINE COMPOUND AND MEDICINAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1995-03-22 EP claimed
US-5616581-A BACTERICIDES YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-04-01 US disclosed
US-5504082-A BACTERICIDE FOR HELICOBACTER, ANTIULCER AGENT, GASTRIC ACIDSUPPRESSOR YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-04-02 US disclosed
EP-0644191-A1 PYRIDINE COMPOUND AND MEDICINAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1995-03-22 EP disclosed