SCHEMBL8916169

SCHEMBL8916169

O=C(O)Cc1cccn2cccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.50
PTGS2 P35354 1/20 0.49
TDP1 Q9NUW8 1/20 0.44
TBXAS1 P24557 1/20 0.42
KDM4E B2RXH2 1/20 0.42
CYP1A2 P05177 1/20 0.42
MAPT P10636 1/20 0.42
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
CYP2C19 P33261 1/20 0.40
CTDSP1 Q9GZU7 2/20 0.40
DUSP3 P51452 1/20 0.40
PTPN5 P54829 1/20 0.40
PTPN11 Q06124 1/20 0.40
BCAT2 O15382 1/20 0.40
NSD2 O96028 1/20 0.39
POLB P06746 1/20 0.39
GRK2 P25098 1/20 0.39
CASP6 P55212 1/20 0.39
CXCL8 P10145 4/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3230868 0.89 AKR1B1 (0.47) AKR1B1PTGS2TDP1KDM4ECYP2C9
SCHEMBL28084372 0.77 ALDH1A1 (0.34) TBXAS1KDM4ECYP1A2MAPTCYP2C9
SCHEMBL24656172 0.74 KDM4E (0.45) AKR1B1PTGS2TDP1TBXAS1KDM4E
SCHEMBL27477607 0.74 TBXAS1 (0.42) PTGS2TDP1TBXAS1KMT2A
SCHEMBL25515799 0.74 APOBEC3G (0.38) TBXAS1KDM4ECYP1A2MAPTHPGD
SCHEMBL12540739 0.73 KDM4E (0.47) AKR1B1PTGS2TDP1TBXAS1KDM4E
SCHEMBL29410826 0.73 AKR1B1 (0.76) AKR1B1PTGS2TDP1KDM4ECYP1A2
SCHEMBL30359 0.73 AKR1B1 (0.76) AKR1B1PTGS2TDP1KDM4ECYP1A2
SCHEMBL28842838 0.71 AKR1B1 (0.73) AKR1B1PTGS2TDP1KDM4ECYP1A2
Hydrochloric Acid SCHEMBL6767821 0.71 AKR1B1 (0.73) AKR1B1PTGS2TDP1KDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113164444-A DOCK1 inhibiting compounds and uses thereof 国立大学法人九州大学 2021-07-23 CN disclosed
US-5674879-A Compositions including and methods of using conformationally restricted angiotensin II antagonist G.D. SEARLE & CO. (US) 1997-10-07 US disclosed