SCHEMBL8916897

SCHEMBL8916897

COc1ccccc1N1CCN(CCC(=O)c2cc3c(s2)CCCC(=O)N3)CC1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 10/20 0.59
ALDH1A1 P00352 2/20 0.54
MAPT P10636 2/20 0.54
KMT2A Q03164 2/20 0.54
ESR1 P03372 1/20 0.54
POLB P06746 1/20 0.54
NR4A1 P22736 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
HTT P42858 1/20 0.52
DRD2 P14416 7/20 0.51
DRD4 P21917 6/20 0.51
DRD3 P35462 6/20 0.51
HTR1D P28221 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8917105 0.95 DRD2 (0.54) HTR1AALDH1A1MAPTKMT2AESR1
Hydrochloric Acid SCHEMBL10838441 0.78 HTR1A (0.65) HTR1AALDH1A1MAPTKMT2APOLB
SCHEMBL8916053 0.77 HTR7 (0.51) HTR1AMAPTKMT2ANPSR1HTT
Hydrochloric Acid SCHEMBL6601969 0.74 HTR1A (0.98) HTR1AALDH1A1MAPTKMT2AHTT
SCHEMBL6352028 0.72 HTR1A (1.00) HTR1AALDH1A1MAPTKMT2APOLB
SCHEMBL20489624 0.72 HTR1A (0.69) HTR1AALDH1A1MAPTKMT2APOLB
SCHEMBL6597937 0.71 HTR1A (1.00) HTR1AALDH1A1MAPTKMT2AHTT
SCHEMBL3254030 0.71 DRD2 (0.63) HTR1ADRD2DRD4DRD3
SCHEMBL10864234 0.71 DRD2 (0.60) HTR1AALDH1A1MAPTKMT2APOLB
Hydrochloric Acid SCHEMBL6598673 0.71 HTR1A (0.98) HTR1AALDH1A1MAPTKMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691330-A ANTIPSYCHOTIC AGENT YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-11-25 US disclosed
US-5532240-A ANTIPSYCHOTIC AGENTS AND ANTISEROTONIN AGENTS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-07-02 US disclosed
EP-0596125-A1 CONDENSED THIOPHENE COMPOUND AND PHARMACEUTICAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1994-05-11 EP disclosed