SCHEMBL8917084

SCHEMBL8917084

COC(=O)c1c(C)nc(N(C(C)=O)C(C)=O)c([N+](=O)[O-])c1-c1ccccc1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LDHA P00338 1/20 0.40
MAPT P10636 6/20 0.39
CYP1A2 P05177 5/20 0.39
CYP2C9 P11712 4/20 0.39
CYP3A4 P08684 4/20 0.39
MEN1 O00255 4/20 0.39
KMT2A Q03164 4/20 0.39
ADORA3 P0DMS8 3/20 0.39
CYP2C19 P33261 3/20 0.39
TSHR P16473 2/20 0.39
NFKB1 P19838 2/20 0.39
CACNA1C Q13936 2/20 0.39
CYP2D6 P10635 2/20 0.39
CRHR1 P34998 1/20 0.38
SMN1; SMN2 Q16637 4/20 0.36
KDM4E B2RXH2 1/20 0.33
RBP4 P02753 1/20 0.32
CLK4 Q9HAZ1 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32
EIF4E P06730 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL904650 0.87 LDHA (0.46) LDHAMAPTCYP1A2CYP2C9CYP3A4
SCHEMBL14941196 0.75 LDHA (0.41) LDHAMAPTMEN1KMT2ACRHR1
SCHEMBL6956083 0.74 MEN1 (0.50) LDHAMAPTMEN1KMT2ASMN1; SMN2
SCHEMBL10763318 0.71 LDHA (0.42) LDHAMAPTMEN1KMT2ASMN1; SMN2
SCHEMBL10745909 0.70 LDHA (0.52) LDHAMAPTMEN1KMT2ASMN1; SMN2
SCHEMBL29351076 0.68 ALDH1A1 (0.48) MAPTCYP1A2CYP2C9CYP3A4MEN1
SCHEMBL744307 0.68 ALDH1A1 (0.48) MAPTCYP1A2CYP2C9CYP3A4MEN1
SCHEMBL11010734 0.68 ALDH1A1 (0.60) LDHAMAPTCYP1A2CYP2C9MEN1
SCHEMBL10745184 0.67 LDHA (0.49) LDHAMAPTSMN1; SMN2KDM4ENPSR1
SCHEMBL6639522 0.67 PDK2 (0.48) MAPTCYP1A2CYP2C9CYP3A4MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5670525-A Substituted 4-phenyl-6-amino-nicotinic acid compounds useful in the treatment of CNS disorders BAYER AKTIENGESELLSCHAFT (DE) 1997-09-23 US disclosed
EP-0705820-A1 6-Amino-nicotinic acid derivatives and their use as selective K-channel modulators BAYER AG (DE) 1996-04-10 EP disclosed