Acridine

Acridine

SCHEMBL8917092

CCCCCCCCCCCCCCCCC(I)CCCCCCCCCN(C)C.c1ccc2nc3ccccc3cc2c1

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 6/20 0.42
DNM1 Q05193 3/20 0.41
ALDH1A1 P00352 1/20 0.41
GLA P06280 1/20 0.41
MAPT P10636 1/20 0.41
HPGD P15428 1/20 0.41
ACHE P22303 1/20 0.41
TRPV1 Q8NER1 5/20 0.39
PPARG P37231 1/20 0.39
PPARA Q07869 1/20 0.39
NPC1 O15118 1/20 0.39
POLB P06746 1/20 0.39
SLC2A1 P11166 1/20 0.39
APOBEC3A P31941 1/20 0.39
RAD52 P43351 1/20 0.39
RAB9A P51151 1/20 0.39
KMT2A Q03164 1/20 0.39
APOBEC3G Q9HC16 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acridine SCHEMBL8920746 0.83 TLR8 (0.44) TLR8ALDH1A1GLAMAPTHPGD
Acridine SCHEMBL8670269 0.83 TLR8 (0.38) TLR8ALDH1A1GLAMAPTHPGD
Acridine SCHEMBL28232031 0.79 ALDH1A1 (0.65) TLR8ALDH1A1GLAMAPTHPGD
Acridine SCHEMBL27681561 0.79 ALDH1A1 (0.65) TLR8ALDH1A1GLAMAPTHPGD
Acridine SCHEMBL28205217 0.77 ALDH1A1 (0.62) TLR8ALDH1A1GLAMAPTHPGD
Acridine SCHEMBL29014290 0.74 ALDH1A1 (0.68) TLR8ALDH1A1GLAMAPTHPGD
SCHEMBL599470 0.72 TLR8 (0.44) TLR8ALDH1A1GLAMAPTHPGD
SCHEMBL20192944 0.72 DNM1 (0.52) DNM1ALDH1A1
Acridine SCHEMBL25416084 0.71 ALDH1A1 (0.54) TLR8ALDH1A1GLAMAPTHPGD
Acridine SCHEMBL8577853 0.71 ALDH1A1 (0.58) TLR8ALDH1A1GLAMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5665328-A USING SELECTED DYE AS BINDING AGENT WITHOUT PRODUCING DETRIMENTAL EFFECT ON MORPHOLOGY OR PHYSIOLOGICAL FUNCTION OF CELLS PHANOS TECHNOLOGIES, INC. (US) 1997-09-09 US claimed
EP-0430968-A4 COMPOUNDS, COMPOSITIONS AND METHOD FOR BINDING BIO-AFFECTING SUBSTANCES TO SURFACE MEMBRANES OF BIO-PARTICLES 1993-10-20 EP claimed
EP-0430968-A1 COMPOUNDS, COMPOSITIONS AND METHOD FOR BINDING BIO-AFFECTING SUBSTANCES TO SURFACE MEMBRANES OF BIO-PARTICLES. ZYNAXIS TECHNOLOGIES INC (US) 1991-06-12 EP claimed
WO-1989010758-A1 COMPOUNDS, COMPOSITIONS AND METHOD FOR BINDING BIO-AFFECTING SUBSTANCES TO SURFACE MEMBRANES OF BIO-PARTICLES ZYNAXIS TECHNOLOGIES, INC. (US) 1989-11-16 WO claimed
EP-0430968-B1 COMPOUNDS, COMPOSITIONS AND METHOD FOR BINDING BIO-AFFECTING SUBSTANCES TO SURFACE MEMBRANES OF BIO-PARTICLES PHANOS TECH INC (US) 1996-11-20 EP disclosed
EP-0430968-A4 COMPOUNDS, COMPOSITIONS AND METHOD FOR BINDING BIO-AFFECTING SUBSTANCES TO SURFACE MEMBRANES OF BIO-PARTICLES 1993-10-20 EP disclosed
EP-0430968-A1 COMPOUNDS, COMPOSITIONS AND METHOD FOR BINDING BIO-AFFECTING SUBSTANCES TO SURFACE MEMBRANES OF BIO-PARTICLES. ZYNAXIS TECHNOLOGIES INC (US) 1991-06-12 EP disclosed
WO-1989010758-A1 COMPOUNDS, COMPOSITIONS AND METHOD FOR BINDING BIO-AFFECTING SUBSTANCES TO SURFACE MEMBRANES OF BIO-PARTICLES ZYNAXIS TECHNOLOGIES, INC. (US) 1989-11-16 WO disclosed