SCHEMBL8917651

SCHEMBL8917651

CCc1c(CCN2CCC(c3noc4cc(O)c(O)cc34)CC2)sc2c1CCN(C(C)=O)C2

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 9/20 0.40
HTR7 P34969 7/20 0.40
DRD2 P14416 4/20 0.40
DRD3 P35462 2/20 0.39
KCNH2 Q12809 5/20 0.39
SLC6A4 P31645 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8917987 0.92 HTR2A (0.49) HTR2AHTR7DRD2DRD3KCNH2
SCHEMBL8918426 0.91 HTR2A (0.44) HTR2AHTR7DRD2DRD3KCNH2
SCHEMBL8917038 0.89 HTR2A (0.50) HTR2AHTR7DRD2DRD3KCNH2
SCHEMBL8918089 0.89 DRD2 (0.54) HTR2AHTR7DRD2DRD3KCNH2
SCHEMBL8917017 0.87 HTR2A (0.46) HTR2ADRD2DRD3KCNH2SLC6A4
Oxalic Acid SCHEMBL8916497 0.87 DRD2 (0.45) HTR2AHTR7DRD2KCNH2
SCHEMBL8916045 0.86 HTR2A (0.36) HTR2AHTR7DRD2DRD3KCNH2
SCHEMBL8917336 0.84 HTR2A (0.44) HTR2AHTR7DRD3KCNH2
SCHEMBL8916743 0.84 HTR2A (0.51) HTR2AHTR7DRD2DRD3KCNH2
SCHEMBL8920271 0.84 DRD2 (0.56) HTR2AHTR7DRD2DRD3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691330-A ANTIPSYCHOTIC AGENT YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-11-25 US disclosed
US-5532240-A ANTIPSYCHOTIC AGENTS AND ANTISEROTONIN AGENTS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-07-02 US disclosed