SCHEMBL8917038

SCHEMBL8917038

CCc1c(CCN2CCC(c3noc4cc(C)ccc34)CC2)sc2c1CCN(C(C)=O)C2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 11/20 0.50
DRD3 P35462 2/20 0.50
DRD2 P14416 8/20 0.44
HTR1A P08908 3/20 0.44
HTR7 P34969 7/20 0.44
KCNH2 Q12809 6/20 0.44
SLC6A4 P31645 2/20 0.43
SLC22A2 O15244 1/20 0.41
CACNA1F O60840 1/20 0.41
ADRB2 P07550 1/20 0.41
CHRM2 P08172 1/20 0.41
CHRM4 P08173 1/20 0.41
CHRM5 P08912 1/20 0.41
ADRA2A P08913 1/20 0.41
CYP2D6 P10635 1/20 0.41
CHRM1 P11229 1/20 0.41
TSHR P16473 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
CHRM3 P20309 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8918426 0.92 HTR2A (0.44) HTR2ADRD3DRD2HTR1AHTR7
SCHEMBL8918089 0.92 DRD2 (0.54) HTR2ADRD3DRD2HTR1AHTR7
SCHEMBL8917017 0.90 HTR2A (0.46) HTR2ADRD3DRD2HTR1AKCNH2
SCHEMBL8917651 0.89 HTR2A (0.40) HTR2ADRD3DRD2HTR7KCNH2
SCHEMBL8917987 0.89 HTR2A (0.49) HTR2ADRD3DRD2HTR1AHTR7
Oxalic Acid SCHEMBL8916497 0.87 DRD2 (0.45) HTR2ADRD2HTR1AHTR7KCNH2
SCHEMBL8920271 0.87 DRD2 (0.56) HTR2ADRD3DRD2HTR1AHTR7
SCHEMBL8917101 0.86 DRD2 (0.54) HTR2ADRD3DRD2HTR7KCNH2
SCHEMBL8916768 0.85 CTSS (0.40) HTR2ADRD3DRD2SLC6A4
SCHEMBL8918706 0.85 DRD2 (0.56) HTR2ADRD3DRD2HTR1AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691330-A ANTIPSYCHOTIC AGENT YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-11-25 US disclosed
US-5532240-A ANTIPSYCHOTIC AGENTS AND ANTISEROTONIN AGENTS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-07-02 US disclosed