SCHEMBL8917674

SCHEMBL8917674

N#Cc1c(-c2ccccc2)nn(-c2ccc([N+](=O)[O-])cc2)c1N

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.58
SMN1; SMN2 Q16637 5/20 0.58
MAPT P10636 4/20 0.58
NPC1 O15118 2/20 0.58
RAB9A P51151 2/20 0.58
NFKB1 P19838 1/20 0.58
NFKB2 Q00653 1/20 0.58
RELA Q04206 1/20 0.58
PKM P14618 2/20 0.50
SRC P12931 1/20 0.50
BRAF P15056 1/20 0.50
KDR P35968 1/20 0.50
LMNA P02545 2/20 0.46
HPGD P15428 2/20 0.46
ADORA2A P29274 1/20 0.46
ADORA1 P30542 1/20 0.46
POLB P06746 2/20 0.46
GAA P10253 1/20 0.45
IKBKB O14920 1/20 0.44
KDM4E B2RXH2 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8309863 0.84 GAA (0.60) ALDH1A1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL8915716 0.78 ADORA1 (0.59) ALDH1A1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL1318935 0.77 IKBKB (0.45) ALDH1A1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL14833516 0.77 BRAF (0.58) ALDH1A1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL8997272 0.77 MAPT (0.44) ALDH1A1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL8309622 0.76 MAPT (0.57) ALDH1A1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL18988429 0.76 ADORA1 (0.56) ALDH1A1SMN1; SMN2MAPTNPC1RAB9A
SCHEMBL8918890 0.75 HTT (0.53) ALDH1A1SMN1; SMN2MAPTLMNAHPGD
SCHEMBL16197283 0.74 BTK (0.48) ALDH1A1MAPTLMNAPOLBIKBKB
SCHEMBL4257428 0.74 IKBKB (0.42) ALDH1A1SMN1; SMN2MAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5593997-A 4-aminopyrazolo(3-,4-D)pyrimidine and 4-aminopyrazolo-(3,4-D)pyridine tyrosine kinase inhibitors PFIZER INC. (US) 1997-01-14 US disclosed