SCHEMBL8915716

SCHEMBL8915716

COc1ccc(-n2nc(-c3ccccc3)c(C#N)c2N)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 7/20 0.59
ADORA2A P29274 6/20 0.59
NPC1 O15118 3/20 0.51
RAB9A P51151 3/20 0.51
HPGD P15428 3/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
POLB P06746 1/20 0.51
CCNA2 P20248 4/20 0.51
CDK2 P24941 4/20 0.51
ADORA2B P29275 3/20 0.50
CDK1 P06493 2/20 0.50
CDK4 P11802 2/20 0.50
CCNB1 P14635 2/20 0.50
CCND1 P24385 2/20 0.50
CDK7 P50613 2/20 0.50
CCNH P51946 2/20 0.50
GAA P10253 1/20 0.50
ALDH1A1 P00352 3/20 0.48
SRC P12931 1/20 0.48
BRAF P15056 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8309863 0.86 GAA (0.60) ADORA1ADORA2ANPC1RAB9AHPGD
SCHEMBL1682478 0.81 LMNA (0.55) ADORA1NPC1RAB9AHPGDSMN1; SMN2
SCHEMBL8309622 0.80 MAPT (0.57) ADORA1ADORA2ANPC1RAB9AHPGD
SCHEMBL14833516 0.79 BRAF (0.58) ADORA1ADORA2ANPC1RAB9AHPGD
SCHEMBL8917674 0.78 ALDH1A1 (0.58) ADORA1ADORA2ANPC1RAB9AHPGD
SCHEMBL18988429 0.77 ADORA1 (0.56) ADORA1ADORA2ANPC1RAB9AHPGD
SCHEMBL8918890 0.77 HTT (0.53) ADORA1ADORA2AHPGDSMN1; SMN2ADORA2B
SCHEMBL8308061 0.77 GAA (0.53) ADORA1ADORA2ANPC1RAB9AHPGD
SCHEMBL11899876 0.76 GAA (0.71) ADORA1NPC1RAB9AHPGDSMN1; SMN2
SCHEMBL14132511 0.76 RAB9A (0.63) ADORA2ANPC1RAB9AHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5593997-A 4-aminopyrazolo(3-,4-D)pyrimidine and 4-aminopyrazolo-(3,4-D)pyridine tyrosine kinase inhibitors PFIZER INC. (US) 1997-01-14 US disclosed