SCHEMBL8918890

SCHEMBL8918890

N#Cc1c(-c2ccccc2)nn(-c2ccc(Cl)c(Cl)c2)c1N

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 4/20 0.53
KDM4E B2RXH2 3/20 0.53
ALDH1A1 P00352 3/20 0.53
GAA P10253 2/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2D6 P10635 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
MAPT P10636 5/20 0.48
TSHR P16473 1/20 0.48
RPA1 P27694 3/20 0.44
ADORA1 P30542 6/20 0.44
ADORA2A P29274 5/20 0.44
ADORA2B P29275 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
LMNA P02545 3/20 0.42
NPSR1 Q6W5P4 2/20 0.42
TDP1 Q9NUW8 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8309863 0.83 GAA (0.60) HTTKDM4EALDH1A1GAAMAPT
SCHEMBL8915716 0.77 ADORA1 (0.59) KDM4EALDH1A1GAAMAPTADORA1
SCHEMBL14833516 0.76 BRAF (0.58) KDM4EALDH1A1GAAMAPTADORA1
SCHEMBL8917674 0.75 ALDH1A1 (0.58) HTTKDM4EALDH1A1GAAMAPT
SCHEMBL8309622 0.75 MAPT (0.57) KDM4EALDH1A1GAACYP1A2CYP2C9
SCHEMBL18988429 0.75 ADORA1 (0.56) KDM4EALDH1A1GAAMAPTADORA1
SCHEMBL8914681 0.72 PLAUR (0.51) HTTKDM4EALDH1A1GAAMAPT
SCHEMBL8915404 0.72 ALDH1A1 (0.49) HTTKDM4EALDH1A1GAAMAPT
SCHEMBL8308061 0.72 GAA (0.53) KDM4EALDH1A1GAAMAPTTSHR
SCHEMBL27847239 0.71 ADORA1 (0.54) HTTKDM4EALDH1A1MAPTADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5593997-A 4-aminopyrazolo(3-,4-D)pyrimidine and 4-aminopyrazolo-(3,4-D)pyridine tyrosine kinase inhibitors PFIZER INC. (US) 1997-01-14 US disclosed