SCHEMBL8309863

SCHEMBL8309863

N#Cc1c(-c2ccccc2)nn(-c2ccccc2)c1N

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.60
ADORA1 P30542 8/20 0.51
ADORA2A P29274 7/20 0.51
ALDH1A1 P00352 6/20 0.50
KDM4E B2RXH2 4/20 0.50
HPGD P15428 3/20 0.50
LMNA P02545 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
MAPT P10636 3/20 0.47
HSD17B10 Q99714 3/20 0.46
ALOX15 P16050 1/20 0.46
MAPK1 P28482 1/20 0.46
MCL1 Q07820 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
TSHR P16473 1/20 0.46
SRC P12931 3/20 0.46
BRAF P15056 2/20 0.46
KDR P35968 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14833516 0.91 BRAF (0.58) GAAADORA1ADORA2AALDH1A1KDM4E
SCHEMBL18988429 0.90 ADORA1 (0.56) GAAADORA1ADORA2AALDH1A1KDM4E
SCHEMBL8309622 0.90 MAPT (0.57) GAAADORA1ADORA2AALDH1A1KDM4E
SCHEMBL8308061 0.86 GAA (0.53) GAAADORA1ADORA2AALDH1A1KDM4E
SCHEMBL8915716 0.86 ADORA1 (0.59) GAAADORA1ADORA2AALDH1A1KDM4E
SCHEMBL8917674 0.84 ALDH1A1 (0.58) GAAADORA1ADORA2AALDH1A1KDM4E
SCHEMBL8918890 0.83 HTT (0.53) GAAADORA1ADORA2AALDH1A1KDM4E
SCHEMBL11546523 0.81 GAA (0.65) GAAALDH1A1KDM4EHPGDLMNA
SCHEMBL8914681 0.81 PLAUR (0.51) GAAADORA1ADORA2AALDH1A1KDM4E
SCHEMBL8915404 0.81 ALDH1A1 (0.49) GAAADORA1ADORA2AALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0745684-B1 Method of quantitative determination of peroxides, a peroxidation-active substance or a pyrazolopyridopyridazine derivative KYOWA MEDEX CO LTD (JP) 1999-08-11 EP disclosed
US-5801008-A Method of quantitative determination of peroxide, a peroxidation-active substance or a pyrazolopyridopyridazine derivative KYOWA MEDEX CO., LTD. (JP) 1998-09-01 US disclosed
US-5593997-A 4-aminopyrazolo(3-,4-D)pyrimidine and 4-aminopyrazolo-(3,4-D)pyridine tyrosine kinase inhibitors PFIZER INC. (US) 1997-01-14 US disclosed
EP-0745684-A1 Method of quantitative determination of peroxide, a peroxidation-active substance or a pyrazolopyridopyridazine derivative KYOWA MEDEX CO., LTD. (JP) 1996-12-04 EP disclosed