SCHEMBL8917774

SCHEMBL8917774

COc1ccc2c(CC3CCN(CCc4c(C)sc5c4CCN(C(C)=O)C5)CC3)noc2c1OC

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 3/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ACHE P22303 2/20 0.34
MAPT P10636 3/20 0.34
ALDH1A1 P00352 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
POLB P06746 1/20 0.34
KDM4E B2RXH2 1/20 0.34
DNMT1 P26358 1/20 0.34
THRB P10828 1/20 0.33
ABCB11 O95342 1/20 0.33
CHRM2 P08172 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33
CHRM1 P11229 1/20 0.33
DRD2 P14416 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
DRD1 P21728 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9411403 0.79 ACHE (0.40) MEN1KMT2AACHEALDH1A1KDM4E
SCHEMBL9411386 0.73 ACHE (0.51) MEN1KMT2AACHE
SCHEMBL9411304 0.71 ACHE (0.45) MEN1KMT2AACHE
SCHEMBL8916147 0.71 DRD2 (0.54) ACHESMN1; SMN2CHRM2HTR1AADRA2A
SCHEMBL8917702 0.70 TP53 (0.39) MEN1KMT2AACHEMAPTSMN1; SMN2
SCHEMBL8917936 0.70 HTR2A (0.53) ACHEALDH1A1SMN1; SMN2CHRM2HTR1A
SCHEMBL9411531 0.69 ACHE (0.63) MEN1KMT2AACHEDRD2DRD4
Fumaric Acid SCHEMBL9411339 0.69 ACHE (0.56) MEN1KMT2AACHEDRD2DRD4
Fumaric Acid SCHEMBL9411345 0.69 ACHE (0.56) MEN1KMT2AACHEDRD2DRD4
SCHEMBL8916687 0.69 DRD2 (0.54) ACHEABCB11CHRM2HTR1AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5691330-A ANTIPSYCHOTIC AGENT YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1997-11-25 US disclosed
US-5532240-A ANTIPSYCHOTIC AGENTS AND ANTISEROTONIN AGENTS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1996-07-02 US disclosed
EP-0596125-A1 CONDENSED THIOPHENE COMPOUND AND PHARMACEUTICAL USE THEREOF YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1994-05-11 EP disclosed